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1-(1-benzofuran-5-carbonyl)-4-[(4-chlorophenyl)methyl]piperazine
8-(2,1,3-benzothiadiazol-4-ylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)sulfamoyl]-N-methylbenzamide
4-(2-fluoro-6-methoxyphenyl)-2-(1,2-oxazol-5-yl)phenol
7-[(2,3-difluorophenyl)methyl]-2-[5-(methoxymethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decane
7-{[(diphenylmethyl)amino]methyl}-5-[(3-fluorophenyl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
8-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-6-amino-2-{2-[(2,3-dimethylphenyl)carbamoyl]acetamido}hexanoic acid
1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)pyrrolidin-2-one
2-(1-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-(furan-2-yl)-2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}propan-1-ol
2-methyl-9-[4-(pyrrolidin-3-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(4-hydroxyphenyl)propyl]acetamide
4-{5-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}pyridine
2-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
(2S,4S)-1-benzyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
7-methyl-3-[2-(3-phenylpiperidin-1-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-ethyl-2-{4-[3-(3-fluorophenyl)benzoyl]piperazin-1-yl}acetamide
(1r,4r)-4-[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]cyclohexan-1-ol
1,3-dimethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
ethyl 1-[2-(cyclohex-1-en-1-yl)acetyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
4-chloro-1,3-dimethyl-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
1-({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)-4-(furan-2-carbonyl)piperazine
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)aniline
dimethyl[1-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)ethyl]amine
1-(2,6-dimethoxypyridin-3-yl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
2-{5-[4-(benzyloxy)piperidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]butan-1-one
methyl 3-[(2-methylpropyl)(pyridin-2-ylmethyl)carbamoyl]propanoate
[(3aS,6aS)-2-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-[5-({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}carbamoyl)pyridin-2-yl]benzoic acid
N-[2-methyl-2-(morpholin-4-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
7-methyl-3-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-N,N-dimethylpiperazine-1-sulfonamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-[(prop-2-en-1-yl)amino]benzamide
1-[1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)ethyl]pyrrolidine
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[1-(pyrazin-2-yl)propan-2-yl]urea
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1-ethyl-1H-1,2,4-triazole
N-{2-[3-(trifluoromethyl)phenyl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(3-carboxy-4-hydroxyphenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylic acid
3-[(3R,4S)-4-(dimethylamino)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-3-yl]propan-1-ol
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(cyclopropylformamido)methyl]benzoate
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1,4-dithiepan-6-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl (2S)-1-{1-[4-(5-phenylpentanamido)phenyl]piperidin-4-yl}pyrrolidine-2-carboxylate
5-{[(5-chlorothiophen-2-yl)methyl]amino}-1-methyl-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4-(thiophene-2-carbonyl)piperazine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(pyridin-4-yl)propanamide
6-methyl-3-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide