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N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,2-dimethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
6-{4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
N-(1,2-diphenylethyl)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
4-{[methyl(oxan-4-yl)amino]methyl}-N-(1-methyl-1H-1,3-benzodiazol-5-yl)benzamide
(3S)-3-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}azepan-2-one
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethylamino)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-methylpyrimidine-5-carboxamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-8-fluoroquinolin-4-ol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-(3-chlorophenyl)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-aminoethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]quinazolin-4-amine
4-(2,5-dimethoxyphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(2,3-dihydro-1H-indol-1-yl)propanoyl]-1-(4-methoxyphenyl)piperazin-2-one
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-azabicyclo[2.2.2]octan-3-amine
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
7-(morpholin-4-ylmethyl)-4-{[4-(pyrrolidin-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(5-chlorofuran-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-3-carbonyl)piperidine
1-ethyl-3-(2-methylpropyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
N,5,7-trimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}-2-[4-(propan-2-yloxy)phenyl]acetic acid
ethyl 1-[(3-hydroxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
7-methoxy-3-{[4-(pyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(4-ethoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
2-benzyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,3-thiazole-4-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(3-hydroxy-3-methylbutyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}benzamide
4-{[5-(4-chlorophenyl)furan-2-yl]methyl}-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 3-[2-(1H-pyrazol-1-yl)acetamido]-5-({[4-(trifluoromethyl)phenyl]formamido}methyl)benzoate
1-cyclopentyl-N-[(3,4-dimethoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,5,7-trimethylquinoline-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[4-(dimethylamino)phenyl]formamido}acetic acid
5-methyl-1-{2-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(morpholin-3-yl)acetamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}ethan-1-one
6-cyclopentyl-2-methoxy-3-[({7H-pyrrolo[2,3-d]pyrimidin-4-yl}amino)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-(1H-imidazol-1-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylbutanamide
3-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl)pyridine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(1S,4S)-2-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
2,3-dimethyl-6-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one