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8-fluoro-3-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-({3-[3-(diethylamino)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
2-[3,5-dimethyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
4-{2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-4-yl)ethyl}morpholine
2-[3-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)phenoxy]acetic acid
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
3-{[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}pyridine
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
2-(3,3-diphenylpiperidin-1-yl)-N-(oxolan-2-ylmethyl)acetamide
6-{[(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)amino]methyl}-1,4-oxazepan-6-ol
3-(1-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
(1R,3S)-3-(2-aminoethoxy)-7-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]pyridine
4-[(4-methoxy-3-methylphenyl)methyl]-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclohexyl-N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
diethyl({1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
5-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
7-hydroxy-4-(2-hydroxy-5-methoxyphenyl)-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
(3R,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,4-dimethylpyrrolidin-3-ol
1-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(3,4-dimethylphenyl)ethan-1-one
(2R,6S)-4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(4-methyl-2-oxopentanoyl)pyrrolidin-3-yl]acetamide
7-{3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carbonyl}-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
2-[9-(3-cyano-6-methylpyridin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
4-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]benzoic acid
2-(2-fluorophenoxymethyl)-N-methyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
[(2S,6S)-4-(1H-imidazol-2-ylmethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
4-{4-[(2,2-diphenylethyl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]propanamide
N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(2-methyl-1-benzofuran-7-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
8-(6-aminopyridine-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3,5-difluoro-2-[2-(3-methoxypropyl)piperidine-1-carbonyl]pyridine
2-(azepan-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)acetamide
5-ethyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
3-(furan-2-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
1-[(5-cyclohexylthiophen-2-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-benzyl-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(2-hydroxyethyl)-2-(5-propylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
{1-[6-(4-fluorophenyl)-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyridin-2-yl]piperidin-3-yl}methanol
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(pyridin-3-ylmethyl)acetamide
3-[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
3-fluoro-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(4-{[2-hydroxy-5-(pyrimidin-2-yl)phenyl]methyl}piperazin-1-yl)ethan-1-one
2-{3-[3-(thiophen-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N,4-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole-5-carboxamide
N-(3,4-dimethoxyphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
2-methyl-N-(1,2-oxazol-3-ylmethyl)-4-phenylpyridine-3-carboxamide
2-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
3-{[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl](methyl)amino}-1λ6-thiolane-1,1-dione