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1-(2-methylpropyl)-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
5-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
4-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(2-hydroxyethyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-1,3-benzodiazole-5-carboxamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
2-{4-[(1-ethyl-1H-imidazol-5-yl)methyl]morpholin-3-yl}acetic acid
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
3-[1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
N,1-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-indole-6-carboxamide
1-(1-cyclohexylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-N4-(furan-2-ylmethyl)piperidine-1,4-dicarboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-cyclopropyl-N-(2-methoxyethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
6-methoxy-3-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-amino-4-(6-ethoxypyridin-3-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(propan-2-yloxy)ethyl]-1,3-oxazole-4-carboxamide
3-{1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
5,8-dimethyl-2-({[3-(morpholin-4-yl)propyl]amino}methyl)quinolin-4-ol
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(4-chloro-2-fluorophenyl)-1-[2-(4-hydroxypiperidin-1-yl)ethyl]urea
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(3-methoxypropyl)piperidine
3,5-dimethyl-1-{3-[2-(2,3,6-trifluorophenyl)-1H-imidazol-1-yl]propyl}-1H-pyrazole
N-[2-(4-chlorophenyl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
N-methyl-3-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]propanamide
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
3-bromo-5-[(furan-2-ylmethyl)sulfamoyl]benzoic acid
1-{2-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
3-cyclopentyl-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-methyl-4-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
4-({3-[(4-chlorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-5-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
3-{[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
3-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-1-methyl-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
methyl (2S)-1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
ethyl 6-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
4-(1H-imidazol-1-yl)-1-[4-(thiophen-2-yl)butanoyl]piperidine-4-carboxylic acid
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
ethyl 2-{1-[(2S,4R)-4-aminopyrrolidine-2-amido]cyclohexyl}acetate
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-methyl-7-(methylsulfanyl)quinoline
N-[1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
5-methyl-N-{[3-methyl-7-(4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}pyrazine-2-carboxamide
6-methoxy-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-4-amine
3-(diethylamino)-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
N-(2-methoxyethyl)-4-[4-(2-methylpropyl)piperazin-1-yl]pyridine-2-carboxamide
N-(3,5-dimethoxyphenyl)-3-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
4-benzyl-1-[3-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
(2R,6R)-4-cyclopentyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{2-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol