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N-{2-[(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidin-6-yl)formamido]ethyl}acetamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]ethan-1-one
1-cyclopentyl-4-[3-(3-propoxypiperidine-1-carbonyl)phenoxy]piperidine
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-4-carbonitrile
7-methyl-2-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
(2R,6R)-4-(3-hydroxypyridine-2-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-[4-(propane-1-sulfonyl)morpholin-3-yl]acetamide
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]thiophene-2-carboxamide
5-[8-methyl-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinolin-2-yl]pyrimidin-2-amine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5,6-dimethylpyridine-3-carboxamide
[(2-tert-butylpyrimidin-5-yl)methyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
4-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
N-[2-hydroxy-1-(thian-4-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
2-[4-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)morpholin-3-yl]acetic acid
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperazine
4-hydroxy-2-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]pyrimidine-5-carboxamide
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)[(3-methyloxetan-3-yl)methyl]amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
ethyl 1-{1-[3-(4-fluorobenzenesulfonamido)phenyl]piperidin-4-yl}piperidine-3-carboxylate
2-(2-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1-methyl-1H-imidazole
N-[3-(dimethylamino)propyl]-2,3,5,6-tetramethylbenzamide
1-(carbamoylmethyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}piperidine-3-carboxamide
1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
9-methoxy-7-(6-methoxypyridazin-3-yl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S)-1,3-dimethyl-4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
N-[(2,6-difluorophenyl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2,6-dimethyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)pyrimidine-4-carboxamide
5-(2-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1,3-dimethyl-1H-pyrazol-5-yl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-(thiolan-3-yl)benzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-ethoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]pyrimidin-2-amine
(2R,3S,6R)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(4-fluorophenyl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]butan-1-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
(3S,4R)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
3-{5-[1-(3,4-dimethylphenoxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-{4-[3-(2H-1,3-benzodioxol-5-yl)propanamido]-2-methoxyphenyl}butanamide
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
5-[4-hydroxy-1-(2-methylbutyl)piperidin-4-yl]-N-methyl-N-(quinolin-5-ylmethyl)-1-benzofuran-2-carboxamide
5-[3-(3-benzoylpiperidin-1-yl)-3-oxopropyl]-5-(2H-1,3-benzodioxol-5-ylmethyl)pyrrolidin-2-one
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine-2-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane