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2-methyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenol
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-yl]propan-1-ol
1-(cyclohexylmethyl)-3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(oxan-4-yl)piperazine
2-{4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazin-1-yl}pyrimidine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
{3-[(2-fluorophenyl)methyl]-1-(3-methylthiophene-2-carbonyl)piperidin-3-yl}methanol
(1R,3S)-7-(4-fluoro-3-methylbenzoyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[1-(methoxymethyl)cyclopentyl]acetamide
(2S,4S)-4-amino-1-{1-[(3,4-dimethylphenyl)amino]cyclohexanecarbonyl}-N-methylpyrrolidine-2-carboxamide
(2S,4S)-1-benzyl-N-ethyl-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N'-[2-(dimethylamino)ethyl]-N-(2-methylphenyl)-N'-[(2-methylphenyl)methyl]propanediamide
4-[4-(furan-3-ylmethyl)piperazin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
5-methyl-5-(4-methylpent-3-en-1-yl)-1-(pyridin-2-ylmethyl)piperidin-2-one
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4,6-dimethylpyrimidine
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
3-(3-chloro-1,2-oxazol-5-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)propanamide
(1R,5R)-6-(cyclopropylmethyl)-3-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-3,4-dimethyl-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-ol
2-(pyridin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
2-methyl-5-({4-[4-(propan-2-yl)piperazine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)-1,3-benzothiazole
({4-cyclopropyl-5-[1-(pyridazin-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
9-methoxy-10-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[methyl(pyridin-2-ylmethyl)amino]-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
1-benzyl-N-[(1-ethylpyrrolidin-3-yl)methyl]-N,2-dimethyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
4-fluoro-N-(2-{[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]formamido}ethyl)benzamide
5-(2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-chlorophenyl)-N-{[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-methyl-2-[3-(1H-pyrazol-3-yl)benzoyl]-1H-imidazole
N-methyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)-N-[1-(pyridin-2-yl)ethyl]propanamide
4-[(dimethylamino)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-ol
1-(3-methylpyridin-2-yl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazine
4-chloro-2-(quinolin-3-yl)phenol
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-oxo-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
N-(4-cyano-2-fluorophenyl)-4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carboxamide
2-({4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)cyclopentanecarboxamide
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenol
2-cyclopropyl-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
[1-(isoquinolin-5-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
[(4-chloro-3-fluorophenyl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-1-carbonyl)-1H-pyrazol-5-amine
3-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,2-diol
N-[2-(5-methylfuran-2-yl)ethyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
4-phenyl-1-(3-propyl-1H-pyrazole-5-carbonyl)-1,2,3,6-tetrahydropyridine
4-{2-[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]ethyl}-3,5-dimethyl-1H-pyrazole
3-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one