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2-(6-oxo-1,6-dihydropyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-N-propyloxane-2-carboxamide
2-benzyl-9-(6-oxopiperazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(2-fluorophenyl)piperidin-4-ol
5-{[4-(2-chlorophenoxy)piperidin-1-yl]methyl}-N-ethylpyrimidin-2-amine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-(5-propyl-1,3,4-oxadiazol-2-yl)-3-(pyrrolidin-1-ylmethyl)piperidine
1,3-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-(1-methoxyethyl)phenyl]-2,5,6-trimethylpyrimidine
N-[(1R,2R)-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]-2,3-dihydro-1H-inden-2-yl]acetamide
2-methoxyethyl 7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
4-[5-fluoro-2-(1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
8-[2-(2-chloro-4-fluorophenoxy)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
3-{[1-(2-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
(3S,4S)-1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
3-[5-(1,1-dioxo-1λ6-thiane-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
1-[4-(dimethylamino)azepan-1-yl]-3-phenoxypropan-1-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
1-{6-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]pyridin-3-yl}ethan-1-one
N-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)methanesulfonamide
N4-{2-[3-(trifluoromethyl)phenyl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(3-cyanophenyl)-3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)urea
(1S,4S)-2-(2-fluorophenyl)-5-[(3-methylquinoxalin-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[7-(4-fluoro-3-methylbenzoyl)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidine
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
9-(cyclopropylmethyl)-1-methyl-4-[3-(pyridin-3-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl]pyridin-2-amine
N-(2-methyl-1-{7-[2-(2-methyl-1H-indol-3-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxolane-3-carboxamide
3-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)thiophene-2-sulfonamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-methoxyethoxy)acetamide
1-(4-cyano-2-ethylphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
N-(2,3-dihydro-1H-inden-1-yl)-5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
9-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
2-(4-cyclopentylpyrimidin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-3-(piperidin-1-yl)propan-2-ol
1-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}-3-(propan-2-yl)urea
1-[2-(1H-imidazol-1-yl)propanoyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-[(1-hydroxycyclohexyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
3-cyclopropyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
4-chloro-5-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(pyrrolidin-1-yl)-1,3-thiazole
N2-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-N4-methyl-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
3-methoxy-1-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one