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(4aS,8aR)-6-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
[(2-chloro-6-fluoro-3-methoxyphenyl)methyl][1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
9-(4-ethoxybenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane
(3R,4R)-4-ethyl-1-(quinoxalin-2-yl)piperidine-3,4-diol
4-(3-{2-azaspiro[4.4]nonane-2-carbonyl}phenyl)-2-methylbutan-2-ol
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-5-phenylpentane-1,5-dione
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]pyridin-2-amine
5-[methyl(2-phenylethyl)amino]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-2,3-dihydropyridazin-3-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-cyclopropyl-6-[(oxolan-2-ylmethoxy)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-N-(1,3-thiazol-2-yl)benzamide
3-[(2-methoxyethyl)sulfamoyl]-N-methyl-N-(oxan-2-ylmethyl)benzamide
methyl 1-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
6-tert-butyl-N-[(1-ethylpiperidin-4-yl)methyl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide
(2S,4R)-N-ethyl-4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
9-hydroxy-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
6-methyl-2-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}ethan-1-ol
N-({1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
4-[3-(2-methylphenoxymethyl)piperidin-1-yl]pyrimidine
7-[2-(2,2,2-trifluoro-1-phenylethoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,4R)-1-[2-chloro-5-(piperidin-1-yl)benzoyl]-3-cyclopropyl-4-methylpyrrolidin-3-ol
6-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
(2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
4-[(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(1S,5R)-6-(2-methoxyethyl)-3-[(2-methoxynaphthalen-1-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
7-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,3-diazepane-2,4-dione
1-[2-(1H-imidazol-1-yl)ethyl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 3-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanoate
ethyl 1-({3-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperidine-2-carboxylate
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-N-ethyl-4-methyl-1,3-thiazol-2-amine
1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyrazin-2-yl)propan-1-one
3-(pyridin-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
N-[1-(3-methylphenyl)piperidin-4-yl]-3-propyl-1H-pyrazole-5-carboxamide
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one
N3-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-3-yl]acetamide
N-[(2,6-difluorophenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
3-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
N-(3-chloro-4-fluorophenyl)-3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide
1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-[2-(1H-imidazol-1-yl)ethyl]-5-[1-(1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(2R,3S)-3-hydroxy-2-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}butanoic acid
N-[2-(1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-4-sulfamoyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide