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N-({3-methyl-7-[2-(phenylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
3-[3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
2-(3-methoxyphenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidine
methyl 2-chloro-5-{[4-(hydroxymethyl)piperidine-1-carbonyl]amino}benzoate
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
4-methyl-5-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
3-[1-(2-amino-4-phenylpyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
N1,N1-dimethyl-N3-[(3-methyl-1-benzofuran-2-yl)methyl]piperidine-1,3-dicarboxamide
2-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-2,3-dihydro-1H-isoindole
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-{[3-(4-propyl-1,4-diazepane-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-methyl-1-phenyl-1H-pyrazole
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(4-fluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-benzyl-3-ethyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
1-(prop-2-en-1-yl)-2-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
2-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-4-carboxamide
6-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-chloro-6-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-3-carboxylic acid
2-[4-(2-ethyl-1-benzofuran-3-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
3-[1-(7-fluoro-2-methylquinoline-4-carbonyl)piperidin-4-yl]phenol
(4aS,7aR)-1-[2-(propan-2-yloxy)acetyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-4-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
8-(5-acetylpyridin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclohexanecarboxamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
methyl 3-{[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]amino}benzoate
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
dimethyl(2-{[(5-methylthiophen-2-yl)methyl](1,3-thiazol-2-ylmethyl)amino}ethyl)amine
1-methyl-2-[1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-ethyl-N-[(1R,2S)-2-phenylcyclopropyl]-1H-indole-5-carboxamide
(1S,3R)-1-[2-(dimethylamino)ethoxy]-N-(3-fluorophenyl)-3-hydroxy-7-azaspiro[3.5]nonane-7-carboxamide
2,3-dimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]quinoxaline-6-carboxamide
2-(pyridin-4-yl)-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidine-5-carboxamide
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-[4-(2-methoxypyridin-3-yl)phenyl]-N-methylacetamide
methyl 5-({2-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]acetamido}methyl)furan-2-carboxylate
1-(2-oxo-2-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}ethyl)pyrrolidin-2-one
N-{[1-(naphthalen-1-ylmethyl)piperidin-3-yl]methyl}ethane-1-sulfonamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
5-phenyl-2-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2H-1,2,3,4-tetrazole
2-(1-cyclopentyl-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
3-(4-chlorophenyl)-4-(3-fluoropyridin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-cyclopentyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide