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methyl (2S,4R)-1-(3-phenylpropyl)-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
(1S,5R)-3-(pyrazin-2-yl)-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-(4-{[1-(6-methoxynaphthalen-2-yl)ethyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
(2-methoxyethyl)[(4-methylphenyl)methyl]{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
5-{1-[(5-ethylpyridin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2-methoxypyrimidine
3-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl}benzoic acid
(3aS,6aR)-5-(1,4-dithiepan-6-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
methyl 2-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}benzoate
1-[3-oxo-3-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propyl]pyrrolidin-2-one
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
3-hydroxy-3-{[(2-methoxyethyl)amino]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
N-[(3R,4R)-3-hydroxy-1-(isoquinoline-3-carbonyl)piperidin-4-yl]pyridine-4-carboxamide
2-benzyl-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-(cyclohex-1-en-1-yl)-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
8-(2-hydroxyethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-[(2,3-dimethoxyphenyl)methyl]-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxypyridin-3-yl)-4-[(1-methoxypropan-2-yl)sulfamoyl]benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-5-ethyl-N-methyl-1H-pyrrole-2-carboxamide
(2E)-3-(3-fluorophenyl)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]prop-2-enamide
6-(2-chlorophenyl)-N-(2-hydroxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1'-[(2-chloro-4-fluorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
(furan-2-ylmethyl)(quinolin-2-ylmethyl)(thiophen-3-ylmethyl)amine
N-butyl-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,3-thiazole-4-carboxamide
N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-3-carboxamide
4-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidin-2-amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(thiophen-3-ylmethyl)propanamide
N-cyclohexyl-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
(pyridin-3-ylmethyl)(quinolin-4-ylmethyl)(thiophen-3-ylmethyl)amine
N-cyclopropyl-1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
3-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2-(pyridin-2-ylsulfanyl)acetamide
2-(2-methoxy-5-methylphenyl)-2-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]acetic acid
N-[4-(morpholin-4-yl)butan-2-yl]-3-propanamidobenzamide
1,3-dimethyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
1-(4-acetyl-1,4-diazepan-1-yl)-3-(2-chlorophenyl)-3-phenylpropan-1-one