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3-{[(2-fluorophenyl)methyl]amino}-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
8-(2-methylfuran-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
ethyl 1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
13-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-(4-{4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl}phenyl)-5-phenylpentanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-ethyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}pyridine
3-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-N,N-dimethyl-1H-1,2,4-triazol-5-amine
1-{4-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]thiophen-2-yl}ethan-1-one
2-(4-fluoro-2-methoxyphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
6-[9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carbonitrile
N1-(3-methylpyridin-2-yl)-N2-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]ethane-1,2-diamine
2-[2-(dimethylamino)ethyl]-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-phenyl-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
1-[(3-fluoro-2-methylphenyl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
(2S)-3-hydroxy-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}propanoic acid
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
N-(6-chloropyridin-3-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
2-(2-aminoethyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}quinazolin-4-amine
1-(3-fluorophenyl)-3-(1-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
methyl 3-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)benzoate
4-(4-chlorophenyl)-N-(1,4-dioxan-2-ylmethyl)butanamide
5-methoxy-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
1-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-(furan-2-ylmethyl)urea
(3S,4S)-1-(1H-imidazol-4-ylmethyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-6-methoxy-1H-indazole
2-(3-ethoxyphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
ethyl 4-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]piperazine-1-carboxylate
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
(2S)-2-amino-N-[2-(2,4-dimethylphenoxy)ethyl]-3-(4-hydroxyphenyl)-N-methylpropanamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-yl)ethan-1-one
1-methyl-3-(3-methylthiophene-2-carbonyl)piperidine
2-{[4-(4-benzyl-5-{[(4-fluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-6-methylpyridine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
4-(4-acetyl-1,4-diazepane-1-carbonyl)-6-ethyl-1,2-dihydropyridin-2-one
({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-ethyl-4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazin-2-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-(1H-imidazol-4-ylmethyl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
2-amino-6-(1H-pyrrol-3-yl)-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
6-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline