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3-[3-(2-methoxyphenyl)phenyl]-1-methyl-1-(1-methylpiperidin-4-yl)urea
2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}-2-[4-(methylsulfanyl)phenyl]acetic acid
1-[3-(1H-pyrazol-1-yl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-amine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
(1R,5R)-6-(cyclopropylmethyl)-3-[2-(4-methylphenoxy)ethanesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-fluoro-3-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]quinolin-4-ol
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-hydroxy-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidine-4-carboxylic acid
(2S,4S)-4-amino-N-[(1S)-2-hydroxy-1-phenylethyl]-1-methylpyrrolidine-2-carboxamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methoxyethoxy)ethan-1-one
1-cyclopropanecarbonyl-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
(2R,6R)-4-[2-(ethylamino)pyrimidine-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-1-yl)phenol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
7-(3-chlorophenyl)-4-[(2-ethylpyrimidin-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N4-(furan-2-ylmethyl)-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
5-methoxy-N,1-dimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
2-{2-[3-(ethylcarbamoyl)pyrrolidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
2-{4-[(3-fluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-(pyridin-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
methyl 9-(4-methanesulfonylpiperazin-1-yl)-3-azaspiro[5.5]undecane-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-(morpholin-4-yl)azetidine-1-carboxamide
2-fluoro-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(benzyloxy)ethyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
(4aS,7aR)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-ethoxy-6-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenol
4-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
8-fluoro-2-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)quinolin-4-ol
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)quinoline-7-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
6-ethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(2,6-dimethoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-pyrazol-5-yl)acetamide
2-[5-(3-acetyl-1H-pyrazol-5-yl)-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl]acetic acid
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-phenoxyphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](2-methoxyethyl)(oxolan-2-ylmethyl)amine
5-cyclopropyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,2-oxazole-3-carboxamide
(4S)-3,3,4-trimethyl-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidin-4-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-(4-fluorophenyl)piperidine