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N-(1-acetylpiperidin-4-yl)-4-(piperidin-3-yl)benzamide
4-methyl-N-[3-(pyridin-2-yl)propyl]-1,3-oxazole-5-carboxamide
4-(1H-pyrazol-1-yl)-1-[3-(thiophen-2-yl)propanoyl]piperidine-4-carboxylic acid
2-[({[1-(ethoxymethyl)cyclopropyl]methyl}amino)methyl]-6-methylquinolin-4-ol
2-{5-[1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)ethyl]-4H-1,2,4-triazol-3-yl}acetic acid
4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
N-(5-acetamido-2-fluorophenyl)-4-(3-methoxypropyl)piperazine-1-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-butyl-N-[(4-fluorophenyl)methyl]acetamide
1-[3-(cyclohexyloxy)-2-hydroxypropyl]-3-(quinolin-6-yl)urea
N,N-dimethyl-5-[(2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamido)methyl]furan-2-carboxamide
(1R,9aR)-1-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}-octahydro-1H-quinolizin-1-ol
N-(1-hydroxybutan-2-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-3-ylmethyl)acetamide
N-(furan-2-ylmethyl)-N,1-dimethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
[2-(7-methyl-1H-indol-3-yl)ethyl][1-(morpholin-4-yl)propan-2-yl]amine
(1R,5R)-3-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-1,3-thiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
6-cyclopentyl-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2,3-dihydro-1H-inden-2-yl)-3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methylpropanamide
2-{4-[2-amino-3-cyano-6-(2-methylbutan-2-yl)pyridin-4-yl]-2-methoxyphenoxy}acetamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
2-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
methyl 6-[(4-benzylpiperidin-1-yl)methyl]-3-cyclopropaneamidothieno[2,3-b]pyridine-2-carboxylate
{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
(1R,3R,5S)-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
8-methoxy-2-[(2-phenylazetidin-1-yl)methyl]quinoline
8-{5-phenyl-1H-pyrazolo[3,4-b]pyridin-6-yl}quinoline
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
1-[1'-(3-chloropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
4-[3-cyclopentyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
3-({1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidin-4-yl}oxy)pyridine
1-(3-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
3-methoxy-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazin-2-amine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
3-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
(3aS,6aS)-2-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(2-methylphenyl)methyl]-3-{2-oxo-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}piperazin-2-one
1-[2-(pyridin-2-yl)ethyl]-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-2-one
1'-(2-methoxypyridine-4-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-methyl-4-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-phenyl-1H-pyrazole
6-{[methyl(pyrazin-2-ylmethyl)amino]methyl}naphthalen-2-ol
2-amino-6-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
2-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}-1-benzofuran-5-carboxamide
5-(4,4-difluoropiperidine-1-carbonyl)-4-propylpyrimidine