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6-{[methyl(2-phenylethyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-2-[({[(2-fluorophenyl)methyl]carbamoyl}methyl)amino]-3-phenylpropanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(1-methoxypropan-2-yl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
1'-(2-hydroxy-5-methylbenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(4,6-dimethylpyridin-2-yl)methyl](methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[1-(thiophen-2-yl)ethyl]pyrrolidin-2-one
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}urea
N-{1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl}acetamide
(4aS,8aR)-6-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
N-{3-[2-(3,4-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}acetamide
2-{[1-(2,3,5,6-tetramethylbenzoyl)piperidin-4-yl]oxy}pyrimidine
N-(2-{1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}quinolin-6-yl)acetamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(piperidin-1-yl)ethan-1-one
4-[(4-fluorophenyl)methyl]-1-(1-methyl-1H-pyrazole-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
methyl 3-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
4-ethyl-3-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2-chlorophenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
5-fluoro-N4,N4-dimethyl-N2-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
N-(butan-2-yl)-5-(methoxymethyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
5-ethyl-1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aR,6aS)-5-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-(2-{4-[2-(2-methylphenyl)acetyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
[(2-chloro-4-fluorophenyl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-cyclopropyl-9-[(3-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-2,1,3-benzoxadiazole
5-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-(2-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}ethyl)-2-methylpropanamide
4-methoxy-3-methyl-N-[(1-methylpiperidin-4-yl)methyl]benzamide
(2S)-N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-dihydro-1H-indole-2-carboxamide
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
1-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-phenoxyethan-1-one
[(3-ethoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
1-(3-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-(2-phenylethyl)-N-(propan-2-yl)cyclohex-3-ene-1-carboxamide
2-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-methoxy-5-{[methyl({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}phenol
1-[4-(oxan-2-ylmethoxy)phenyl]-3-(pyridin-3-ylmethyl)urea