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N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]-4-oxoadamantane-1-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-ethyl-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidin-4-amine
5-acetyl-N,2,4-trimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrrole-3-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(morpholin-4-yl)ethan-1-one
N-(2-{1-[(3-methylphenyl)methanesulfonyl]piperidin-2-yl}ethyl)acetamide
2-ethyl-8-[2-(2-fluorophenyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[3-(pyrrolidin-1-yl)phenyl]methyl}urea
2-amino-6-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
2-(azocan-1-ylmethyl)-4-hydroxyquinoline-6-carboxamide
4-(hydroxymethyl)-1-[3-(hydroxymethyl)quinolin-2-yl]piperidin-4-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclohexanecarboxamide
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
[(3R,4R)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-(3-fluorophenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
N3-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}piperidine-1,3-dicarboxamide
(2S,4R)-4-(3,4-difluorobenzamido)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrrolidine-2-carboxamide
1,3,6-trimethyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
5-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-phenyl-1H-1,2,3,4-tetrazole
N-(4-fluorophenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
2-(2-{1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,2-oxazole-4-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
N-(2,2-difluoroethyl)-4-{[(5-methyl-1H-pyrazol-3-yl)methyl]sulfamoyl}benzamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(5-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[4-(5-oxo-5-phenylpentanoyl)morpholin-3-yl]acetamide
N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(quinoline-6-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 3-[({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}carbamoyl)amino]propanoate
2-amino-4-[2-(furan-2-yl)phenyl]-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
3-(2-{[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]formamido}acetamido)propanoic acid
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-[4-(2-phenylethyl)piperazin-1-yl]-6-(piperidine-1-carbonyl)pyrazine
9-(furan-2-carbonyl)-1-methyl-4-(2-phenylpropyl)-1,4,9-triazaspiro[5.5]undecane
2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
5,6-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]acetamide
1-[4-(3-methylphenoxy)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
4-(1H-imidazol-1-ylmethyl)-1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-ol
3-phenyl-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[(2R,3R)-1'-(1H-1,3-benzodiazole-5-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-{4-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
methyl (1R,3S,3aR,6aS)-3-(2-fluoro-4-methylphenyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-({1-[(4-fluorophenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl}methyl)acetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(5-propyl-1,3,4-thiadiazol-2-yl)-decahydroisoquinoline