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5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
1-(2-aminoethyl)-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-(1H-indol-2-ylmethyl)-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
9-(1,4-dioxan-2-ylmethyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4,6-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-amine
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
3-{[4-(2-methoxy-3,5-dimethylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-N,N-dimethylbenzamide
{[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}(methyl)(pyridin-4-ylmethyl)amine
N-[2-(1H-imidazol-4-yl)ethyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(5S,9aS,9bS)-5-(isoquinolin-5-yl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
1-cycloheptyl-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
5-methyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]phenol
N-(2-methoxy-5-methylphenyl)-2-{[4-(methylamino)pyrimidin-2-yl]amino}acetamide
1-[2-(dimethylamino)-4-{[3-(1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[1-(pyrimidin-4-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
ethyl 4-{methyl[1-(pyridin-4-yl)ethyl]amino}piperidine-1-carboxylate
2-(2-methoxyethyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
2-phenyl-N-[3-(propan-2-yloxy)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-(2-methylphenoxy)-1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
2-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
methyl 9-(cyclopentyloxy)-7-oxo-3-(1,3-thiazole-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[3-(2-methoxyphenoxy)propyl]pyridine-4-carbonitrile
N-{1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pyrrolidin-3-yl}acetamide
1-ethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)-1H-pyrrole
1,9-dimethyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-chlorophenyl)-4-(5-phenyl-1,3-oxazole-4-carbonyl)morpholine
9-(3-ethyl-1,2-oxazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}thiophene-2-carboxamide
N-ethyl-5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}pyrimidin-2-amine
N-[(2R,3R)-2-methoxy-1'-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(3-methylcinnolin-5-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]acetamide
2-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-1,2,3,4-tetrahydroisoquinoline
2-amino-4-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
2-(6-aminopyridin-3-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
N-benzyl-1-cyclopropyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-6-(1H-pyrazol-1-yl)pyrimidine
2-(2,3-dihydro-1H-isoindol-2-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
6-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
(8R,9aS)-2-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
5-ethyl-1'-(quinoline-8-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,9aR)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(3-{[2-(2-hydroxyethoxy)ethyl]sulfamoyl}benzoyl)piperidine-3-carbonitrile