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1-(4-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
8-(3-methyl-1,2-oxazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
(1R,5R)-3-benzoyl-6-[2-(benzyloxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
2-(2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethoxy)ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-methyl-1-[4-({2-[(2-methylquinolin-8-yl)oxy]ethyl}amino)piperidin-1-yl]propan-1-one
1-(2-methylphenyl)-3-(1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-(6-methoxypyridin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1S,5R)-3-(oxan-4-yl)-6-[(3,4,5-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(methylamino)-N-[3-(2-phenylacetamido)phenyl]benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidin-3-yl]methanol
(1S,3R)-3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]cyclohexan-1-amine
1-(2-methoxy-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
3-(2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
3-(2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-[4-({1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-1,2,3-triazole
methyl 4-methyl-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzoate
3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)urea
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(3-methylphenyl)piperidine
3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
5-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-5-oxopentanamide
1-(2-methyl-5-sulfamoylphenyl)-3-[(2-propyl-1,3-thiazol-4-yl)methyl]urea
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}acetamide
3-(2-hydroxypropan-2-yl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-(1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}azetidin-3-yl)-1H-pyrazole
7-methoxy-3-{[methyl(thian-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]cyclohexanecarboxamide
1-{1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}piperidin-4-ol
2-[(2,2,6,6-tetramethylpiperidin-4-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(5-methylpyrazin-2-yl)methyl]-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-[4-(methylsulfanyl)phenyl]urea
(1R,5S,6R,7S)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,3-dimethyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-{[5-(2-fluorophenyl)furan-2-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1-(trifluoromethyl)cyclopropane-1-carboxamide
N,6-dimethyl-2-(piperidin-1-yl)-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)cyclohexyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-(2-propoxyethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-benzyl-4-[4-(1,2,4-oxadiazol-3-yl)pyridin-2-yl]piperazin-2-yl}ethan-1-ol