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5-(3,3-diphenylpiperidine-1-carbonyl)-2-methyl-3,4-dihydropyrimidin-4-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethylfuran-3-carboxamide
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
(3S,4S)-1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-methylpiperidine-3,4-diol
(2S,4S)-4-amino-1-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrrolidine-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
2-(butylsulfanyl)-5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
(3S,4R)-1-(2-methoxypyrimidine-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-(2-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}ethyl)-2-methylfuran-3-carboxamide
2-methyl-N-{[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}propanamide
3-(2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
3-{[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}-1-methyl-1H-indole
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-ethoxy-1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-[(3R,4S)-1-(4-chloro-3-methylbenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
4-(benzyloxy)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
5-benzyl-5-{1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-methyl-N-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1S,5R)-3-benzyl-6-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-chloro-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-amino-N-(2,1,3-benzoxadiazol-5-ylmethyl)cyclopropane-1-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(2S,6S)-4-[4-(trifluoromethyl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-(4-{3-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-ol
1,5-dimethyl-4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[2-(azepan-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(3aS,6aS)-2-({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-3-(2-methylpropyl)-N-(4H-1,2,4-triazol-4-yl)-1H-pyrazole-5-carboxamide
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(thiophene-2-sulfonyl)pyrrolidine-2-carboxamide
2-(3-methoxyphenyl)-N,N-dimethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonamide
1-{[1-(quinoline-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
9-(2-methoxybutanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3,5-dimethyl-7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
1-methyl-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[3-(methylsulfanyl)phenyl]methyl}urea
9-[(2-fluoro-3-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}-1H-indole
1-(4-methoxybenzoyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine
[2-ethoxy-5-({[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]methanol
8-(4-methyl-1H-pyrrole-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1S,5R)-3-(5-fluoro-2-methoxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-methyl-1-[1-(pyridin-4-yl)piperidin-4-yl]butan-1-ol