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5-({2-[(dimethylamino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
methyl N-{2-[3-(2-methylphenoxy)azetidin-1-yl]-2-oxoethyl}carbamate
ethyl 4-[6,7-dimethoxy-3-({[(3S)-2-oxoazepan-3-yl]amino}methyl)quinolin-2-yl]piperazine-1-carboxylate
1-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-4-(4-methoxyphenyl)piperazine
2-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[(cyclopropylmethyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
ethyl 5-[6-amino-5-cyano-4-(oxolan-3-yl)pyridin-2-yl]-2-methylfuran-3-carboxylate
1-[(4aR,8aR)-7-[(4-fluoro-3-methoxyphenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
7-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(furan-2-ylmethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
N-ethyl-3-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4,5-dimethylthiophen-2-yl)methyl]piperidin-3-ol
4-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-one
4-ethyl-3-{1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[8-(4-chloro-2-fluorobenzoyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
methyl (2S,4S)-1-(naphthalen-1-ylmethyl)-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
ethyl 4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine-1-carboxylate
N-(2H-1,3-benzodioxol-5-yl)-7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecane-3-carboxamide
3-chloro-N-(2-methoxyethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
9-[(2S)-2-amino-3-hydroxypropanoyl]-2-(thiophen-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3-(5-{1-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-2-yl)propanamide
2-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane
2-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-[1-(thiophen-2-yl)butyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
7-methoxy-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-3-carboxamide
1-({5-[1-(cyclopentylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(1-methyl-1H-indol-4-yl)methyl]piperidin-4-ol
N-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-1H-indazole-3-carboxamide
N4-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
N-[(3-methylphenyl)methyl]-5-(1,4-oxazepane-4-carbonyl)-1-propyl-1H-1,3-benzodiazol-2-amine
2-(2-aminoethyl)-N-[2-(2-ethoxyphenyl)ethyl]quinazolin-4-amine
1-(azepan-1-yl)-2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
2-(piperidin-1-yl)-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}acetamide
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-2-(4-chlorophenyl)acetic acid
8-fluoro-2-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}quinolin-4-ol
(4aS,8aR)-6-(pyrazin-2-yl)-1-(1,3-thiazol-2-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-{[5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]methyl}pyridine
4-ethyl-3-{1-[3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one