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(1,4-dioxan-2-ylmethyl)[(6-ethoxyquinolin-2-yl)methyl]methylamine
1-[2-(2-methyl-1H-indol-3-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
4-(2-amino-3-cyano-6-cyclobutylpyridin-4-yl)benzamide
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine
ethyl 4-[5-(cycloheptylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carbonyl]piperazine-1-carboxylate
4-({3-[(4-methoxyphenyl)methyl]-1-phenyl-1H-1,2,4-triazol-5-yl}methyl)piperazin-2-one
ethyl 2-({7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecane-3-carbonyl}amino)propanoate
2-(2-chlorophenoxy)-N-[(3-methylpyridin-4-yl)methyl]acetamide
N-[3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]-3-methoxybenzamide
N-(9H-fluoren-9-yl)-1-{2-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
2-amino-4-(3-chloro-4-propoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[3-(3-fluorophenyl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
5-(1H-imidazol-2-ylmethyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-methyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
6-[(3-methoxyphenyl)methoxy]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-(morpholin-4-yl)-2-{3-[(thiolan-3-yl)amino]phenoxy}ethan-1-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-(4,6-dimethylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-N-[2-(pyridin-3-yloxy)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
dimethyl(3-{2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-[2-(azepan-1-yl)-2-oxoethyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(3-methoxyphenyl)amino]-N-methylbutanamide
(3aS,6aS)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-N-methyl-1,3-thiazol-2-amine
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl}pyrazine-2-carbonitrile
2-methoxy-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[(4,5-dimethylfuran-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
3-({4-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
2-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[1-(morpholine-4-sulfonyl)piperidin-3-yl]-3-phenylpropan-1-one
1-(furan-2-ylmethyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
4-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
1-methyl-2-oxo-8-(1,3-thiazol-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N,N-dimethylpyrrolidin-3-amine
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine
7-(3-chlorophenyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-hydroxycyclohexyl)methyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)carbamoyl)butanoate
3-(2-methoxyphenyl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
N3-[4-(3-methoxyphenyl)phenyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-(2-methoxyethyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-(cyclopropylmethyl)-4-phenylmethanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(1H-pyrazol-4-yl)butanamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[2-(methylsulfanyl)ethyl]piperazine
N-(2-methoxyethyl)-2-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
2-(1-methyl-1H-imidazol-2-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
7-chloro-2-methyl-4-[4-(2-propoxyethyl)piperazine-1-carbonyl]quinoline
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(3-hydroxyphenyl)ethan-1-one
1-[3-(3-ethylphenoxy)azetidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one