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[2-(4-phenyl-1H-imidazol-1-yl)phenyl]methanol
N3-(2-methylpropyl)-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-ethoxy-6-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}phenol
N-[(4-methylphenyl)methyl]-2-(thiomorpholin-4-ylmethyl)quinazolin-4-amine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-(pyridin-2-yl)piperazine
(3aS,6aS)-2-cyclopentanecarbonyl-5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-ethyl-5-methyl-N4-[3-(4-methylpiperazin-1-yl)propyl]pyrimidine-2,4-diamine
(2S,4S)-4-amino-1-(2,1-benzoxazole-3-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
2-[6-chloro-3-(1H-imidazol-2-yl)imidazo[1,2-a]pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]azonan-2-one
3-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
3-({2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
(4aS,7aR)-1-[2-(1H-imidazol-1-yl)acetyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-[1-(3-methylbutyl)-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl]ethan-1-ol
4-(2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepane-1-carbaldehyde
3-{[(1H-indol-2-ylmethyl)amino]methyl}-1-(2-methoxyethyl)-6-methyl-1,2-dihydroquinolin-2-one
N-{[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
2-[4-(hydroxymethyl)phenyl]-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
1-(3,4-dichlorophenyl)-5-[2-(1H-imidazol-1-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-phenyl-3-(pyridin-2-yl)propanamide
1-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
6-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2,4-dimethylpyridine-3-carbonitrile
N-ethyl-6-(2-fluoro-4-methoxyphenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-1-methylpiperazin-2-yl)methanol
1-[(2-methoxyethyl)carbamoyl]-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
7-(cyclobutylmethyl)-2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(pyrimidine-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1H-1,3-benzodiazol-2-yl)-2-{methyl[(5-phenyl-1H-pyrazol-4-yl)methyl]amino}acetamide
2-acetyl-8-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[methyl(2-phenylethyl)amino]-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[(2-fluorophenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-cyclohexyl-3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]propanamide
3-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
8-(piperidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-[1-(methylsulfanyl)propan-2-yl]-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-4-(2-oxopyrrolidin-1-yl)butanamide
2-{4-[4-(difluoromethoxy)benzoyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
methyl 6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridine-3-carboxylate
3-[(oxan-4-yl)sulfamoyl]-N-(pyridin-2-ylmethyl)benzamide
1-ethyl-4-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidin-2-one
2-(3-methoxypropyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-4-methanesulfonyl-2-[(2,3,6-trimethylquinolin-4-yl)formamido]butanoic acid
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine