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1-(2-{[(furan-2-ylmethyl)(prop-2-yn-1-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
(4aR,8aR)-2-cyclobutanecarbonyl-7-[2-(2-methoxy-4-methylphenoxy)ethyl]-decahydro-2,7-naphthyridin-4a-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
2-[2-hydroxy-2-(thiophen-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,5R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
5-(2,4-difluorophenoxymethyl)-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[3-(azepane-1-carbonyl)phenyl]-1-[1-(pyrazin-2-yl)propan-2-yl]urea
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-[2-(2,4-difluorophenyl)-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
3-phenyl-5-(4,4,4-trifluorobutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclohexylacetamide
(3S,7S)-5-(2-methyl-1H-pyrrole-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanamido)acetic acid
2-amino-4-(1,5-dimethyl-1H-indol-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,5S)-5-[3-(piperidin-1-yl)azetidine-1-carbonyl]pyrrolidin-3-amine
N,N-dimethyl-2-[(1S,5R)-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
1-(azocan-1-yl)-3-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-(1-hydroxy-2-methylpropan-2-yl)-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
7-(6-methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
1-[6-(dimethylamino)pyrimidin-4-yl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-({[3-(4-hydroxyphenyl)propyl]amino}methyl)piperidin-3-ol
(3R,4R)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
N-(pentan-3-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)pyridine
1-[1-(5-phenoxyfuran-2-carbonyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-{5-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-(1-ethylpiperidin-4-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
N-{4-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutyl}acetamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
(1R,9aR)-1-(1H-1,2,4-triazol-1-ylmethyl)-octahydro-1H-quinolizin-1-ol
1-ethyl-6-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide
2-(2-methoxyethyl)-8-[2-(methylsulfanyl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N-diethyl-7-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane-2-carboxamide
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-[(4aR,8aR)-7-[2-(3-chlorophenyl)acetyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
2-[1-(3-methanesulfonylbenzoyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
1-(2-methoxy-5-methylbenzenesulfonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-[4-(4-benzylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
N-[2-(1H-imidazol-1-yl)ethyl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-(2-ethoxyethyl)-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
1-(4-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}phenyl)imidazolidine-2,4-dione
N-[(5-methoxy-1H-indol-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide