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5-chloro-3-methyl-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]-1H-indole-2-carboxamide
2-[(dimethylamino)methyl]-4-({2-methyl-2,8-diazaspiro[4.5]decan-8-yl}methyl)phenol
methyl 3-({2-[(4-chlorophenyl)methyl]-1,3-benzoxazol-5-yl}formamido)propanoate
4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
ethyl 1-(cyclopropylmethyl)-5-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1r,4r)-4-{[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]methyl}cyclohexane-1-carboxylic acid
3,3-dimethyl-1-[(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
2-{4-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
7-(cyclohexylmethyl)-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decane
2-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxan-4-amine
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-{4-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]piperidin-1-yl}prop-2-en-1-one
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-(thian-4-yl)piperazine
ethyl 1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidine-3-carboxylate
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
methyl 3-methoxy-5-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carbonyl}benzoate
2-[4-(1H-imidazol-1-yl)phenyl]-1-[(2S)-oxolan-2-ylmethyl]-1H-imidazole
1-[5-(ethanesulfonyl)thiophen-2-yl]-1H-indazole
1-(furan-2-ylmethyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2R,3R,6R)-5-(2-cyclopropylpyrimidine-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[1-(but-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]propan-2-yl}furan-2-carboxamide
2-(pyridin-2-yl)-5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-1-yl}-4,6-dimethylpyrimidine
3-(2-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}ethyl)-4-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(1H-indol-1-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4R)-1-(cyclopent-1-ene-1-carbonyl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
2-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
3-[(dimethylamino)methyl]-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-ol
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(3R,5R)-N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-phenylpropanamide
3-methyl-8-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(4-fluorophenyl)methyl]methylamine
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
{4-[5-(1-methyl-1H-imidazol-5-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
methyl 3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
1-(furan-2-ylmethyl)-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
(4aR,8aR)-2-(pyrrolidine-1-carbonyl)-7-(quinolin-5-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
N-methyl-N-[2-(oxan-2-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(2S,4S)-4-amino-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[5-(7-fluoro-3-methyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(morpholin-4-yl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
6-(1-{1-[(4-methylphenyl)amino]cyclopentanecarbonyl}piperidin-3-yl)pyrimidin-4-ol
2-methyl-8-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[4.5]decane