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[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
N-(3-chloro-4-methoxyphenyl)-3-{1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}propanamide
4-({[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2,6-dimethoxyphenol
2-({4-[4-(2-amino-1H-imidazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
2-{4-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-(cyclohexylmethyl)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N4-methyl-N4-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
4-(4-chlorophenoxy)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
(3S,9aR)-3-propyl-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,9aR)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-octahydro-1H-quinolizine-1-carboxamide
2-(1,3-thiazol-2-yl)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[1-(1-hexylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
3-(2-methoxyethyl)-5-(1-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
(3R,4R)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
N,3,6-trimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-benzofuran-2-carboxamide
methyl 2-(2,3-dihydro-1-benzofuran-5-yl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxylate
4-methoxy-N-(1-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-8-fluoroquinoline
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[(3R,4S)-1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(furan-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-1-(4-methylphenyl)piperazin-2-one
7-[(6,8-dimethyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(butylsulfanyl)-6-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]pyrimidin-4-amine
5-(1-cyclohexanecarbonylpiperidin-4-yl)-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[3-(furan-2-yl)phenyl]piperidin-4-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,4-diazepane
5-[2-(benzylamino)ethyl]-1-[2-(3-methoxyphenyl)ethyl]pyrrolidin-2-one
1-methyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-methyl-2-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
14-[4-(1H-1,2,4-triazol-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-ethyl-2-{4-[(3-fluoropyridin-4-yl)methyl]piperazin-1-yl}-N-methylpyrimidin-4-amine
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
(2S,4R)-4-(benzylamino)-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
(2S)-2-hydroxy-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenylethan-1-one
4-[(8-fluoroquinolin-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
6-(3-chlorophenyl)-2-[2-(hydroxymethyl)piperidine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(3-methoxyphenyl)-3-methyl-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
(2S,4R)-4-[(naphthalen-1-ylmethyl)amino]-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
8-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[(4-fluorophenyl)methyl]-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide