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N-cyclopropyl-3-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
1-(2,3-dimethylphenyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
2-[1-(3,5-dimethylphenyl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
1'-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[4-(isoquinolin-5-yl)phenyl]-2-methylpropanamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(phenylsulfanyl)acetamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
N-(1-carbamoylcyclopentyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
2-{5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-2,2-diphenylacetamide
(2S)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-hydroxy-2-phenylethan-1-one
4-({3-[2-(2-ethylphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)benzoic acid
(3R,4R)-1-{[2-(furan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
7-(3-methoxypropyl)-2-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-3-carboxamide
(1R,5S,6S)-3-[2-methyl-2-(piperidin-1-yl)propyl]-N-[(1r,4r)-4-hydroxycyclohexyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-[(3R,4S)-1-[(2,5-dimethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
7-(2-methoxyethyl)-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(furan-2-ylmethyl)amino]-N-(2-hydroxyethyl)-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]furan-2-carboxamide
4-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2,5-dimethylpyrimidine
N-methyl-4-{12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}benzene-1-sulfonamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methanol
4-[2-(pyrrolidin-3-yl)benzoyl]-1λ6-thiomorpholine-1,1-dione
3-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}pyridine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-[(3-fluorophenyl)methyl]piperidine-1-carboxamide
2,3-dimethyl-6-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-ethyl-1-(3-methylbutyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
5-ethyl-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine
2-(4-{[4-(furan-2-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1-benzyl-N3-ethyl-N5-[2-(4-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
dimethyl(1-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}ethyl)amine
(1S,5R)-3-[2-(methylamino)pyridine-4-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{1-[(3,5-difluorophenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
3-{5-[(2S)-2-hydroxy-2-phenylacetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(2-hydroxyethyl)propanamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
2-[N-(3-fluorophenyl)methanesulfonamido]-N-methyl-N-(1H-pyrazol-5-ylmethyl)acetamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(prop-2-en-1-yl)piperazine
(2S)-2-{4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}-3-(4-hydroxyphenyl)propanoic acid
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
7-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-[(3,4-dimethylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-{[(2-ethyl-6-methylpyridin-3-yl)oxy]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
N-(1H-imidazol-2-ylmethyl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-ethyl-N-[1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine