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(4-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
4-{[N-ethyl-3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}benzoic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
N-butyl-N-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
N-(dicyclopropylmethyl)-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
N-(2-{[1-(2-methoxyethyl)pyrrolidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-3-ethylpiperidin-3-yl}methanol
N-cyclopropyl-1-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-fluorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
(3S,4S)-4-(piperidin-1-yl)-1-[(2,4,6-trimethoxyphenyl)methyl]pyrrolidin-3-ol
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
7-[(2R)-oxolane-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
(1S,6R)-9-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[4-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]acetic acid
N-(2-hydroxyethyl)-3-{5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-phenylethyl)piperidine-3-carboxamide
2-{[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-[(prop-2-en-1-yl)amino]benzamide
1-(6-aminopyrimidin-4-yl)-4-benzyl-1,4-diazepan-6-ol
N-(butan-2-yl)-N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-(3-chloro-2-fluorophenyl)-1-methyl-1-(thian-4-yl)urea
6-[(3,5-dimethoxyphenyl)methoxy]-4-(1-methyl-1H-indole-2-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
7-(3,6-dimethylpyrazin-2-yl)-4-(3-fluoropyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1,3-benzoxazol-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
3-(3-amino-5-fluoro-1H-indazol-1-yl)-5-(azepane-1-sulfonyl)benzoic acid
4-methyl-N-[2-methyl-5-(2-propanamidopropanamido)phenyl]benzamide
2-(2-methoxyphenoxy)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}acetamide
3-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1-methylpiperidine-2-carboxamide
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-3,5-difluoro-N-[(2-methylphenyl)methyl]pyridine-2-carboxamide
2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}morpholine
1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(2-methylphenyl)-4-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-yl)piperazine
2-(dimethylamino)-4-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
N-{4-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]phenyl}acetamide
(3aR,6aS)-5-(cyclohexylcarbamoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}benzamide