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1-[3-(cyclohexylsulfanyl)propyl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
8-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-methoxy-1-{1'-[2-(3-methylphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-(2-methoxyethyl)-3-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}propanamide
4-[2-(propanamidomethyl)phenyl]benzamide
methyl({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N,N-dimethyl-4-(1-methyl-1H-indole-6-carbonyl)piperazine-1-sulfonamide
1-{1-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}piperidin-4-ol
4-hydroxy-2-(pyridin-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
2-methoxy-3-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrazine
2-(dimethyl-1,2-oxazol-4-yl)-5,8-dimethoxy-4-methylquinoline
4-acetyl-N-[2-chloro-5-(morpholin-4-yl)phenyl]-1,4-diazepane-1-carboxamide
ethyl (4aS,8aR)-6-(4-methoxypyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylate
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(4-propanoylphenoxy)acetamide
4-chloro-1,5-dimethyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
14-heptyl-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(2-phenylethyl)-4-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}benzamide
(1R,5R)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(4aS,8aR)-6-[(3,5-dimethoxyphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-chloro-2-methyl-6-(2,3,4-trimethoxyphenyl)pyrimidin-4-ol
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-[(3-methoxyphenyl)amino]-N-methyl-N-(quinolin-8-ylmethyl)butanamide
1-[(4-methylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)acetyl]piperazin-2-one
2-hydroxy-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-4-(methylsulfanyl)butanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-{5-[(methylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazole
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(5-methylfuran-2-yl)methyl]amino}pyrrolidin-2-one
(butan-2-yl)[(2-chlorophenyl)methyl]{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}amine
2-(1H-imidazol-2-yl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]benzamide
3-fluoro-4-[4-(piperidine-1-carbonyl)phenyl]pyridine
8-methoxy-5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]quinoline
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-ethylpyrimidine
1-ethyl-6-methyl-N-[(1-methylpiperidin-4-yl)methyl]-2-oxo-N-(2-phenylethyl)-1,2-dihydropyridine-3-carboxamide
N-cyclopropyl-2-(2-oxoimidazolidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1,3-dimethyl-6-(pyridin-2-yl)-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4-phenyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine-4-carbonitrile
4-ethyl-1-methyl-3-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,3-dihydro-1H-isoindole-2-carbonyl)-6-(2,5-dimethylfuran-3-yl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
2-acetamido-3-hydroxy-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
5-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
6-cyclopropyl-2-[4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
[5-({4-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)furan-2-yl]methanol
[3-(1H-imidazol-1-yl)-1-phenylpropyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyloxan-4-amine
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
1-methyl-3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-{3-[3-(5-chloro-2-hydroxyphenyl)-1H-pyrazol-1-yl]phenoxy}acetic acid
1-(3-benzoylpiperidin-1-yl)-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(3R,4R)-1-[1-(2-fluorophenyl)piperidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol