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5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazole
1-(benzenesulfonyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
ethyl 2-(1-{2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamido}cyclohexyl)acetate
6-(3-methoxypiperidin-1-yl)-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-{[(propan-2-yl)({[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
1-(6-methoxyquinolin-8-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
ethyl 3-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]amino}propanoate
(4-{[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}phenyl)urea
N-(butan-2-yl)-5-(methoxymethyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
1-[(6-methylpyridin-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(5-{[1-(2,5-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-4H-1,2,4-triazol-3-yl)ethan-1-amine
N-(2-fluorophenyl)-3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}propanamide
2-chloro-6-methoxy-3-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}phenol
1-(2,5-dimethylfuran-3-carbonyl)-3-(1H-imidazol-2-yl)piperidine
(2R,6R)-4-[2-(4-fluoro-3-methylphenyl)acetyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
1-methyl-3-{[4-(morpholine-4-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(4aS,8aS)-N-[4-chloro-3-(dimethylcarbamoyl)phenyl]-4a-hydroxy-decahydroisoquinoline-2-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-1,3-benzodiazole
N-cyclopropyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(thiophen-3-ylmethyl)acetamide
4-[4-(1H-pyrazol-3-yl)phenyl]piperidin-4-ol
N-(4-fluoro-3-methylphenyl)-4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
1-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(1,2,3-thiadiazol-5-yl)urea
3-{5-cyclopentyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[2-(dimethylamino)ethyl]propanamide
4-(2-butylpyrrolidine-1-carbonyl)-2-(2,3-difluorophenoxymethyl)-1,3-oxazole
3-(1-methoxyethyl)-4-(naphthalen-1-yl)-4H-1,2,4-triazole
3-phenoxy-N-[1-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
4-[4-(1-ethyl-3-methylpiperidine-3-carbonyl)piperazin-1-yl]-6-methylpyrimidin-2-amine
3-[2,5-difluoro-4-(trifluoromethyl)phenyl]-1-[3-(morpholin-4-yl)propyl]urea
3-[1-(cyclohex-1-en-1-yl)ethyl]-1-{3-[(dimethylsulfamoyl)amino]phenyl}urea
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(3,3,4-trimethylpiperazin-1-yl)butan-1-one
3-(2-chloropyridin-3-yl)-1-(2-methylpropyl)-1-(pyridin-4-ylmethyl)urea
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-2-(2-oxopyrrolidin-1-yl)propanamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
9-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}(propan-2-yl)amine
N-methyl-4-[(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)sulfamoyl]thiophene-2-carboxamide
3-(7-hydroxy-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1-propylpiperidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-{1-oxaspiro[4.5]decan-3-yl}acetamide
1-[(2S)-1-cyclohexanecarbonylpyrrolidine-2-carbonyl]-4-(1H-imidazol-2-yl)piperidine
2-[({4-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)sulfanyl]pyridine
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(2S)-2-amino-N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(1H-imidazol-4-yl)propanamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(1-benzofuran-2-ylmethyl)pyrrolidin-3-yl]-4-methylpiperazine