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5-phenyl-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]pentan-1-one
1-(cyclopropylmethyl)-N-ethyl-5-{[3-(2-methylphenyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-3-methylbenzoic acid
8-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-amino-1-{3-[(3-hydroxyphenyl)carbamoyl]propanoyl}-N-methylpyrrolidine-2-carboxamide
(4aS,8aR)-1-butyl-6-(2-ethoxypyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 3-{[1-(2-methoxyethyl)-4-oxo-5-{[(1-phenylcyclopentyl)methyl]carbamoyl}-1,4-dihydropyridin-3-yl]formamido}propanoate
(3S,4R)-3-ethyl-4-methyl-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-ol
N-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]-3-oxopropyl}acetamide
(3aR,6aR)-2-[4-(1H-imidazol-1-yl)butanoyl]-5-(propan-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(phenylsulfanyl)propyl]imidazo[1,2-a]pyrimidine-2-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-2-methylpyridine
N-[(3S,4R)-1-[(3-methylthiophen-2-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-tert-butyl-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-methyl-2-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}aniline
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-amino-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
N-[(3S,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-({2,5-dimethyl-3-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)-1,2-dimethylpiperazine
N-ethyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydroquinazoline-2-carboxamide
2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
5-(2,5-dimethylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(4-{2-[(dimethylamino)methyl]phenyl}phenyl)acetamide
1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-3-amine
2-amino-6-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
7-fluoro-3-{[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(2,3-dimethylphenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-amine
N-{2-[2-(hydroxymethyl)phenyl]phenyl}cyclopropanecarboxamide
1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
methyl 1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-3-carboxylate
4-{1-[1-(2-methoxyacetyl)piperidine-4-carbonyl]piperidin-3-yl}benzoic acid
(3S,5S)-1-[(3-chlorophenyl)methyl]-N-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
2-[2-(dimethylamino)ethyl]-8-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,7aR)-1-[(3,5-difluorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,7aR)-1-(2,4-dimethoxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
7-[(3,4-difluorophenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-ethyl-1-(6-methylpyridin-3-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]urea
2-{4-chloro-2-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}acetic acid
2-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidine-3-carbonyl)pyridine
2-[9-(2,5-dimethylfuran-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
(3R,4R)-1-cycloheptanecarbonyl-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-methylazepane-2-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
5-[5-(ethylsulfanyl)thiophen-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{methyl[(2-phenylphenyl)methyl]amino}propanamide