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N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-amino-6-benzoyl-4-(3-ethyl-1,2-oxazol-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
1-(3-methoxyphenyl)-4-[2-(2-methyl-1H-indol-3-yl)acetyl]piperazin-2-one
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
1'-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)spiro[indene-1,4'-piperidine]
3-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
ethyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
4-hydroxy-2-(4-methylphenyl)-N-[(6-methylpyridin-2-yl)methyl]pyrimidine-5-carboxamide
1-{[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)acetamide
N-methyl-2-{2-[2-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}pentanamide
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
N-methyl-5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)furan-2-carboxamide
5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(oxan-4-yl)pyrrolidin-3-yl]acetamide
5-benzyl-4-(3-hydroxypropyl)-1-(3-methoxyphenyl)piperazin-2-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-methoxy-N-(2-methoxyethyl)-2-{[1-(2-methylpropanoyl)piperidin-4-yl]oxy}benzamide
3-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
(3aR,6aR)-2-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-(cyclopropylsulfamoyl)-6-[2-(naphthalen-2-yl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(2-fluorophenyl)methyl]-1-[(2S)-1-(piperidin-4-yl)pyrrolidine-2-carbonyl]piperidine
2-(dimethylamino)-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
N-(1-methyl-1H-pyrazol-4-yl)-2-[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]acetamide
2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-[(2-methylphenyl)methyl]acetamide
2-[2-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}amino)phenyl]-N,N-dimethylacetamide
(2S,4S)-4-amino-N-(2-methoxyethyl)-1-methyl-N-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-(2-methylnaphthalen-1-yl)-5-oxopyrrolidine-3-carboxylic acid
4-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-4-oxobutane-1-sulfonamide
(1R,7S)-N-(furan-2-ylmethyl)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(pyrrolidin-1-yl)benzamide
4-(1-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-4-yl}ethyl)morpholine
N-{2-[(1-methyl-1H-1,3-benzodiazol-5-yl)formamido]ethyl}pyridine-3-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
(3S,4S)-3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-4-hydroxy-1λ6-thiolane-1,1-dione
3-[1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1,3-oxazolidin-2-one
3,5-dimethyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-4-sulfonamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-oxo-2-(pyridin-3-yl)acetamide
1-(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)pyrrolidin-2-one
3-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(1,2,3-thiadiazol-5-yl)urea
(1R,3S)-3-methoxy-7-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
2-(3-chloro-4-hydroxyphenyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(4aS,7aR)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(3-methylphenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one