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[(5-chloro-2-ethoxyphenyl)methyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
(benzylsulfamoyl)(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
4-[6-(pyridin-4-yl)pyridine-3-carbonyl]morpholine
N-({7-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
7-(5-chloropyridin-2-yl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(propan-2-yloxy)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
methyl(oxan-2-ylmethyl)[(2,3,4-trimethoxyphenyl)methyl]amine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
3-[1-(3,5-dichloro-4-methylbenzoyl)azetidin-3-yl]pyridine
3-cyclopropyl-1-(4-methanesulfonylphenyl)-5-(3-methylfuran-2-yl)-1H-1,2,4-triazole
2-(azepan-1-yl)-1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)ethan-1-one
2-cyclopropyl-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrimidine-5-carboxamide
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
4-(3-chlorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrimidin-2-amine
3-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole
1-(1H-1,3-benzodiazole-5-sulfonyl)-1,4-diazepan-6-ol
5-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}phenyl)pyrrolidin-2-one
(3aR,6aS)-5-[4-(1H-imidazol-1-yl)benzoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-chlorophenyl)-4-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-5-methyl-1,3-oxazole
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(1,2,4-oxadiazol-3-yl)piperidine
1-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidin-3-ol
1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(2-phenoxyethyl)-1,4-diazepan-5-one
4-ethyl-6-[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]pyrimidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
5-(3-acetylphenoxymethyl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
methyl 4-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-hydroxypyrazine-2-carboxamide
(1S,6R)-9-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(2S,3S)-2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-methylpentanamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}amine
3-{2-[5-(3,4-dichlorophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
5-tert-butyl-2-[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]-1H-1,3-benzodiazole
3-{[1-(2-methylpropanoyl)piperidin-3-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-(5-acetamido-2-methylphenyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
methyl 3-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethoxy}benzoate
7-(3-chlorophenyl)-4-(2-hydroxybutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-[3-(dimethylamino)phenyl]-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
2-cyclopropyl-8-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
4,5-dimethyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)pyrimidine
N-(5-chloro-2-methoxyphenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
(3S,7S,8aS)-7-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3aR,6aS)-5-{[2-(benzyloxy)phenyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
4-({5-[2-(5-methylfuran-2-yl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)pyrimidine
5-(methoxymethyl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]furan-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}piperidin-2-one
3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea