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[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidine-3-carboxylate
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-imidazole
4-({2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-(2,2-dimethyloxan-4-yl)-1-[2-(propan-2-yloxy)ethyl]-1H-1,2,3-triazole
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methyl-1H-pyrrole-3-carboxamide
[(2S,6S)-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-(1-methyl-5-oxopyrrolidin-3-yl)urea
4-[(2-methoxyphenyl)methyl]-11-[(2-phenylethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(1H-pyrazol-1-yl)-N-[2-(thiophen-2-yl)ethyl]benzamide
6-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(morpholin-4-yl)pyrimidin-4-amine
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pent-4-enamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(3S,9aR)-2-methyl-3-(2-methylpropyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N3-(furan-2-ylmethyl)-N5-[2-methyl-2-(morpholin-4-yl)propyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclohexyl-5-[2-(1H-imidazol-2-yl)phenyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
[(3R,5S)-1-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-5-(hydroxymethyl)piperidin-3-yl]methanol
6-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxamide
4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(3-fluorophenyl)-1H-pyrazole
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-methyl-2-(6-methylquinolin-5-yl)pyridine-3-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrrole-2-carboxamide
4-methoxy-N-({1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-3-(3-methylthiophene-2-carbonyl)piperidine
1-cyclopentyl-4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-methyl-2-(2-{[2-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-1-phenylmethanesulfonamide
1-ethyl-4-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine
5-cyclopropanecarbonyl-1'-(3,5-difluoropyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
6-chloro-2-{[4-(thian-4-yl)piperazin-1-yl]methyl}quinoline
{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
8-methoxy-5-[5-(pyrrolidine-1-carbonyl)furan-2-yl]quinoline
ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2-methoxyethyl)piperidine-3-carboxylate
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
[1-(2,5-dimethylbenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
4-acetyl-N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanamide
3-cyclopropyl-4-[(1S)-1-phenylpropyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-fluoro-N-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]benzamide
2-[(3-fluorophenyl)methyl]-6-methyl-3-(4-methylpiperazine-1-carbonyl)-1-[3-(morpholin-4-yl)propyl]-1,4-dihydropyridin-4-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide