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N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridazine-4-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}acetamide
5-fluoro-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-methyl-6-oxo-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,6-dihydropyrimidine-5-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]quinoline-6-carboxamide
4-(5-chlorothiophen-2-yl)-7-(2-methoxyethoxy)-1,2,3,4-tetrahydroquinolin-2-one
(4aR,7aS)-1-acetyl-4-(1H-indole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4R)-1-(5-chloro-2-methoxybenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenol
9-(3-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 1-(but-2-ynoyl)-4-(2-phenylethyl)piperidine-4-carboxylate
5-methyl-1'-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-5-(1,2,5-trimethyl-1H-pyrrol-3-yl)-1H-imidazole
4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
4-{[5-(1-cyclopropanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(3-methylbut-2-en-1-yl)amine
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(1H-indol-3-yl)acetamide
4-(4-fluorophenyl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
1-(4-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-ethyl-N-(pyridin-4-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-ethyl-3-[(2-fluorophenyl)formamido]-N-(oxan-4-ylmethyl)propanamide
1-[(2,4-dimethoxyphenyl)methyl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1H-imidazole-5-carboxamide
2-tert-butyl-5-(4-methyl-1,4-diazepane-1-carbonyl)pyrimidin-4-ol
2-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)-N-methylacetamide
2-(2-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
7-[(2,3-difluorophenyl)methyl]-2-(6-methoxypyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{[(2-methoxypyrimidin-5-yl)methyl](pyridin-3-ylmethyl)amino}butan-1-ol
2-{5-[(adamantan-1-ylsulfanyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
[(3R,4R)-1-(2-methoxy-4-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3aR,6aR)-2-(2-chlorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)pyridin-2-amine
1-ethyl-4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-(2-methyl-1H-imidazol-1-yl)-1-[4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(2S,4R)-1-[(3-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)acetamido]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2,2-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}oxane-4-carboxamide
6-methyl-2-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(1S,5R)-3-[2-(2-chloro-4-methylphenoxy)ethyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 6-(2-methylpropyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate