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2-methyl-6-[1-(thiophene-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
8-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-(4-{[1-(2,5-dimethylfuran-3-yl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}acetic acid
3-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[(4aR,7aS)-4-[(6-methylpyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aR,7aS)-1-ethyl-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methylphenyl)methyl]-N-[1-(4-methylphenyl)propyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5S,6R)-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-{1-[1-(2,2-difluoroethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
ethyl 1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(1-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-({[(2-ethylpyrimidin-5-yl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-methoxypropanamide
5-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(3-fluoro-4-phenylbenzoyl)piperidine
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(pyridin-4-yl)propanamide
2-({4-[2-(dimethylamino)benzoyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-5-(naphthalen-2-yl)-1,2,4-triazine
N-[(3-methylpyridin-4-yl)methyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
7-[(3,4-difluorophenyl)methyl]-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-(1H-indazol-6-yl)-3-methylurea
2-(4-hydroxypiperidin-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N-methyl-N-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}thian-4-amine
2-{3-[1-(dimethylamino)ethyl]phenyl}benzamide
(3S,4S)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(propan-2-yloxy)pyrrolidin-3-ol
(1R,5S)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-benzyl-3-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-methyl-1,4-diazepan-5-one
(1S,6R)-9-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
11-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
(1S,4R)-4,7,7-trimethyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carboxamide
2-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)propanamide
8-methyl-2-propyl-N-[2-(thiophen-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-(pyridin-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
2-ethyl-7-methoxy-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
3-(3,4-difluorophenyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
2-amino-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide