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1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
5-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
(3S,7S,8aS)-7-{[(3,4-dimethylphenyl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
7-cyclohexyl-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
5-[1-(3,5-dimethyl-1H-pyrazol-4-yl)propan-2-yl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2-fluorophenoxymethyl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
3-[2-(4-hydroxypiperidin-1-yl)ethyl]-6-methoxy-3,4-dihydroquinazolin-4-one
N-{[2-(butan-2-yloxy)phenyl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
5-(5-ethyl-1,3-oxazole-4-carbonyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1R,5R)-6-(2-methoxyethyl)-N-[4-(methylsulfanyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-chloro-3-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
1-acetyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
(1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
5-amino-4-chloro-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carboxamide
1-methyl-N-[(1-methylpiperidin-3-yl)methyl]-6-oxo-N-(2-phenylethyl)-1,6-dihydropyridine-3-carboxamide
(1H-imidazol-2-ylmethyl)(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[1-(1-cyclohexanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
8-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[2-(dimethylamino)ethyl]-6-methyl-N-[(5-methylthiophen-2-yl)methyl]pyridine-2-carboxamide
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
4-fluoro-3-[3-(3-methylphenoxy)azetidine-1-carbonyl]benzene-1-sulfonamide
3-ethyl-6-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1,3-benzoxazol-2-one
4-(2-{3-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)benzene-1-sulfonamide
2-methyl-N-({3-methyl-7-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}pyridin-1-ium-1-olate
dimethyl({[6-(3,4,5-trimethoxyphenyl)pyridin-3-yl]methyl})amine
1-cyclopropyl-5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]piperidin-2-one
(1R)-2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylethan-1-ol
4-[(3-fluorophenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
(4aS,7aR)-1-(1-methyl-1H-imidazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,7aR)-5-methyl-2-(2-methyl-2-phenoxypropanoyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-[3-fluoro-5-(2-methylpropoxy)phenyl]-4-methoxybenzamide
2-({4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-5-ethyl-1,3,4-thiadiazole
4-(5-ethylfuran-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
ethyl 4-(3-phenylpropyl)-1-(propane-1-sulfonyl)piperidine-4-carboxylate
4-[2-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)phenyl]morpholine
2-(1H-1,3-benzodiazol-1-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
6-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[1-(2-benzyl-1,3-thiazole-4-carbonyl)azetidin-3-yl]pyridine
(3S,4S)-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}propanamide
6-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}pyridine-2-carboxylic acid
4-fluoro-N-{2-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide