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3-[(4-methyl-6-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}pyrimidin-2-yl)amino]phenol
N-[2-(dimethylamino)ethyl]-5-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-N,2,2-trimethyloxan-4-amine
6-[methoxy(phenyl)methyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[2-(2,4-dimethylphenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
1-[(2-methoxyphenyl)methyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
5-methyl-3-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-1H-indole
5-butyl-4-(2-methanesulfonylacetyl)-1-(3-methylphenyl)piperazin-2-one
1-(2-methoxyphenyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
N-({5-[(2,3-difluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
ethyl 1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
1-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]ethane-1-sulfonamide
N-cyclopropyl-3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(1-methoxybutan-2-yl)quinoxaline-5-carboxamide
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperidin-4-yl]acetamide
(2S,4R)-4-butanamido-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-methyl-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
N,N-dimethyl-4-[({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]benzamide
2-(methylsulfanyl)-5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azocane
2-[4-(hydroxymethyl)phenyl]-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
7-(1,3-benzothiazol-2-yl)-4-[(5-chloro-2-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[hydroxy(pyridin-2-yl)methyl]-N-(2-methyl-1-benzofuran-5-yl)piperidine-1-carboxamide
2-(1-ethylpiperidin-4-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
9-(2-phenylacetyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-1-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
methyl 4-{[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
methyl(oxolan-3-ylmethyl)(quinoxalin-2-ylmethyl)amine
2-[2-(2,2-dimethylmorpholin-4-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
3-[(2R,3R,6R)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,6-dihydroxy-N-methylbenzamide
2-{4-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-1-yl}-N-ethylacetamide
4-[(4-{4-oxo-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}phenyl)methyl]-1λ6-thiomorpholine-1,1-dione
6-(azepan-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
4-ethyl-2-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
2-(oxan-2-ylmethoxy)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-[2-(dimethylamino)ethyl]-N-methyl-5-oxo-N-(1H-pyrazol-3-ylmethyl)pyrrolidine-3-carboxamide
N,4-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
7-(cyclopropylmethyl)-2-{2-[4-(methylsulfanyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
methyl 4-(5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2,4-oxadiazol-3-yl)benzoate
N5-cyclopropyl-N6-{[1-(morpholin-4-yl)cyclopentyl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-{4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
1-[cyclohexyl(methyl)amino]-3-[4-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine