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[(1-methyl-1H-imidazol-2-yl)methyl][(2-methylphenyl)methyl](prop-2-en-1-yl)amine
1-[1-(5-chloropyridine-2-carbonyl)piperidin-4-yl]piperidin-3-ol
5-(2-chlorophenyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)furan-2-carboxamide
5-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-methoxypyrimidine
N-methyl-2-[3-oxo-1-(2,7,8-trimethylquinoline-4-carbonyl)piperazin-2-yl]acetamide
N-methyl-2-propyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyridine-4-carboxamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
N-cyclopentyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
3-(3-fluorophenyl)-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one
4-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[1-(propan-2-yl)-1H-pyrazol-4-yl]piperidine-1-carboxamide
1-ethyl-5-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}pyrrolidine-3-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[(4-methylphenyl)methyl]piperidine
N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
4-({2-[1-(naphthalene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
6-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]pyridine-2-carboxylic acid
2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
3-(3-hydroxy-3-methylbutyl)-N-[(4-hydroxyphenyl)methyl]benzamide
1-[2-(furan-2-ylmethoxy)phenyl]-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N,N,5-trimethylpyrimidin-4-amine
3-(2,6-dimethoxypyridin-3-yl)-2-methyl-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
(3S,4S)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
2-(5-chloro-2-methoxyphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
2-({[2-(furan-2-yl)-2-hydroxyethyl]amino}methyl)-6,8-dimethylquinolin-4-ol
5-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-(4-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
N-[(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(4-phenylmethanesulfonylmorpholin-3-yl)acetic acid
N,N,4-trimethyl-5-[4-(2-phenylethyl)piperazine-1-carbonyl]pyrimidin-2-amine
4-[2-(benzyloxy)acetyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
1-{[(2S,4S)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-fluoropyrrolidin-2-yl]methyl}-3,3-dimethylurea
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]propanamide
(3S)-1-(dimethyl-1,3-thiazole-5-carbonyl)-N,N-dimethylazepan-3-amine
1-[1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)cyclopentanecarboxamide
5-{[2-(2-methylphenyl)-1H-imidazol-1-yl]methyl}-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidin-2-amine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
2-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}-4H-chromen-4-one
3-(2-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)pyridine
N-[(3R,4R)-1-(5-cyanopyridin-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
4-({2-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}methyl)morpholine
(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
1-(2-{[(2-chloropyridin-3-yl)methyl](methyl)amino}pyrimidin-4-yl)pyrrolidin-3-ol
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)propan-1-one