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5-ethyl-1'-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[1-(1H-imidazol-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-N-methylthiophene-2-carboxamide
4-(3-chlorophenoxy)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
7-methyl-3-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
1-{4-[4-(1-methylpiperidine-2-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
5-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[(4-methylpiperidin-1-yl)sulfonyl]pyrrolidin-3-yl]acetamide
3-[3-(furan-2-yl)-1H-pyrazol-1-yl]-5-(morpholine-4-sulfonyl)benzoic acid
3-(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
8-(3-methoxybenzenesulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(4aS,7aR)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
2-methyl-N-(2-{[2-(2-oxopiperidin-1-yl)ethyl]carbamoyl}phenyl)furan-3-carboxamide
9-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(4-methylphenoxymethyl)furan-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(2-chlorophenyl)-4-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-one
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-7-azaspiro[3.5]nonan-1-ol
3-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)-3,9-diazaspiro[5.6]dodecan-10-one
3-cyclopentyl-1-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)urea
(1S,5R)-3-benzyl-6-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
4-(cyclopropylmethyl)-1-[2-(3,4-dimethylphenoxy)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(cyclopropylmethyl)-N-methyl-5-[2-(1,3-thiazol-4-yl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-5-carboxamide
3-phenyl-8-[4-(1H-pyrazol-4-yl)butanoyl]-1,8-diazaspiro[4.5]decan-2-one
N-[3-methyl-2-(pyrrolidin-1-yl)butyl]-5-propyl-1,3,4-oxadiazol-2-amine
3-[(dimethylamino)methyl]-1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
2-methoxyethyl N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamate
2-[4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)piperidin-1-yl]acetic acid
4-[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-methanesulfonyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
2-(4-chlorophenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
N-cyclopentyl-5-[(4-methoxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,2S,6R,7S)-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
N-(1-{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)acetamide
ethyl 4-[6-(1H-1,3-benzodiazol-2-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
methyl 8-[(4-methoxynaphthalen-1-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 4-({[(3R,5S)-5-(ethylcarbamoyl)-1-(1-propylpiperidin-4-yl)pyrrolidin-3-yl]amino}methyl)benzoate
1-{4-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
3-[(4aR,7aS)-6,6-dioxo-4-(pent-2-yn-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-[(2-cyclohexyl-1H-imidazol-1-yl)methyl]pyridine
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-2-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-4-acetamido-N-(furan-2-ylmethyl)benzamide
3-[1-(2,3-dihydro-1H-inden-4-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]propanamide
3-(4-chlorobenzoyl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine