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N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
3-chloro-5-fluoro-N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}benzamide
3-(1H-1,3-benzodiazol-2-yl)-1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridazin-3-amine
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-5-tert-butyl-1,3,4-oxadiazol-2-amine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-benzyl-8-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-2-hydroxypyridine-3-carboxamide
2-[2-(benzyloxy)phenyl]-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
(1-{[2-(difluoromethoxy)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]piperidin-3-yl)methanol
N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
5-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-phenyl-1H-imidazole-4-carboxamide
4-{2-cyclohexyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
9-(4-methoxypyrimidin-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
6-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
1-(3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3,5-dimethyl-2-[4-(oxolane-2-carbonyl)-1,4-diazepane-1-carbonyl]-1H-indole
methyl 4-({4-[4-(methoxycarbonyl)phenyl]piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
1-methyl-9-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-[(2-fluorophenyl)methyl]-3-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-chloro-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-fluorobenzamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
4-{2-[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
3-{1-[1-(3-chlorophenyl)piperidin-4-yl]piperidin-3-yl}-N-cyclopropylpropanamide
6-(3-methoxypyrazin-2-yl)quinoline
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]quinoline
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(quinolin-2-ylmethyl)-1,4-diazepan-2-one
(4aS,7aR)-1-(4-fluoro-2-methylbenzenesulfonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
N-(3-methyl-4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)acetamide
{4-[4-(4-fluorophenyl)oxane-4-carbonyl]-1,4-oxazepan-6-yl}methanol
4-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-1λ6-thiane-1,1-dione
4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-(propan-2-yl)piperidine
9-(2-hydroxypyridine-3-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(cyclohexylmethyl)-4-[(6-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl]ethan-1-ol
2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-amino-8-(1-benzofuran-2-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
6-[(4aR,8aS)-6-(4-phenylbutanoyl)-decahydro-1,6-naphthyridine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
4-ethyl-3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1,4-diazepane-1-carbonyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzene-1-sulfonamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
methyl 2-[butyl(methyl)sulfamoyl]-6-[(4-acetamidophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-methoxy-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(2-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-2-yl}ethyl)pyridine