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3-{5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(2-hydroxyethyl)propanamide
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
6-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,2-benzoxazole
1-(ethanesulfonyl)-3-(2-phenylethyl)piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2,5-dihydro-1H-pyrrole-2-carboxamide
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
4-ethoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-[1-(methoxymethyl)cyclopentyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
8-chloro-2-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}quinolin-4-ol
4-(5-fluoro-2-methylphenyl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-fluorophenyl)methyl]-4-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
2-methoxy-5-({[2-(pyrrolidin-1-yl)ethyl]carbamoyl}amino)benzamide
methyl 2-(pyrrolidine-1-sulfonyl)-6-(quinoxaline-6-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-ethyl-3-[(1-{2-[(propan-2-yl)amino]benzoyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(3-ethynylbenzoyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-(morpholin-4-yl)azetidine-1-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-(1H-indazol-1-yl)-N-methylacetamide
1-(cyclopropylmethyl)-4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-(propan-2-yl)-1,4-diazepane
(1-{[(5-tert-butyl-1,3,4-oxadiazol-2-yl)(methyl)amino]methyl}cyclobutyl)methanol
(benzylsulfamoyl)({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine
3-(cyclopentylsulfamoyl)-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
ethyl[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]{[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
1-(1-cyclohexylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N4-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methyl-1,3-thiazol-2-amine
methyl 4-methyl-3-({[2-(propylsulfanyl)ethyl]carbamoyl}amino)benzoate
3-(3-hydroxy-3-methylbutyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-cyclopropyl-N-({2-[methyl(thiophen-3-ylmethyl)amino]-7-(methylsulfanyl)quinolin-3-yl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2-methoxy-5-methylphenyl)formamido]-N,N-dimethylbutanamide
N'1-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N'1-(oxolan-2-ylmethyl)cyclopropane-1,1-dicarboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
2-cyclopropyl-4-hydroxy-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrimidine-5-carboxamide
3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propane-1,2-diol
1-(2,3-dihydro-1H-indol-1-yl)-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-oxopiperazine-1-carboxamide
4-{2-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}morpholine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}ethan-1-one
3-{4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-1-yl}benzoic acid
1-(4-fluoro-2-methylphenyl)-3-[4-(oxolan-2-yl)butyl]urea
5-({[2-(azepan-1-yl)ethyl](methyl)amino}methyl)pyrimidin-2-amine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
2-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(5-hydroxy-1,2-dimethyl-1H-indol-3-yl)formamido]-N,4-dimethylpentanamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-cyclobutyl-1H-1,2,4-triazol-3-yl}acetamide
1-(azepan-1-yl)-3-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1,3-dimethylpiperazin-2-one