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1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(thian-4-yl)piperazine
2-methoxy-1-{3-[4-(pyridin-3-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)pyridin-2-amine
N-({3-methyl-7-[4-(thiophen-2-yl)butanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
N-methyl-3-(N-methyl-1-2,3,4,9-tetrahydro-1H-carbazol-8-ylformamido)butanamide
(2E)-3-(2-chlorophenyl)-N-cyclopentyl-N-({4-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)prop-2-enamide
3-chloro-5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-methoxy-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methylbenzamide
N-[4-(furan-2-yl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxamide
4-methanesulfonyl-2-[(3-methoxyphenyl)methyl]morpholine
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
(1R,7S)-3-cycloheptyl-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(2-ethoxyethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(4-hydroxyphenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
N-[3-({[(1S)-1-carbamoyl-3-methylbutyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
4-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-pyrazol-1-yl)propan-1-one
(1S,5R)-3-[(1-methyl-1H-indol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
N-(2-methoxyethyl)-1-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(2R,4R)-N-[(1R)-1-(4-fluorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide
(2R,6R)-11-methoxy-4-(3-propyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3R,4R)-4-amino-1-[2-(2-fluorophenyl)benzoyl]piperidin-3-ol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
4-{[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1,2-oxazole
3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-methoxyphenyl)urea
(2S,4R)-4-cyclopropaneamido-N,N-diethyl-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
5-{4-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
2-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-[(2-fluorophenyl)methyl]acetamide
2-(adamantan-1-ylformamido)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
2-methyl-5-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
methyl 2-(ethylsulfamoyl)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3-methoxyphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
1-(5-ethylthiophene-3-carbonyl)-3-(2-methylphenoxy)azetidine
2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)pyridine-3-carbonitrile
1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}piperazine
N-(1,2-oxazol-3-ylmethyl)-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylic acid
methyl 4-[2-amino-3-cyano-6-(2,4-difluorophenyl)-5-methylpyridin-4-yl]-1H-pyrazole-3-carboxylate
N-(furan-3-ylmethyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-4-methyl-1H-imidazole-5-carboxamide
1-methyl-3-{[2-(trifluoromethoxy)phenyl]methyl}imidazolidin-2-one
2-{[4-(prop-2-en-1-yl)piperazin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(4-hydroxyphenyl)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
5,6-dimethyl-N-[2-(morpholin-4-yl)butyl]pyrimidin-4-amine