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1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(5-fluoro-2-methylphenyl)methyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N-cyclopropyl-1-(5-hydroxypyrazine-2-carbonyl)piperazine-2-carboxamide
1-methyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine-2-carboxylic acid
N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-cyclohexyl-1-phenyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4,6-dimethyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
4-(cyclohex-3-en-1-yl)-1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole
2-ethyl-9-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(piperidin-1-ylmethyl)benzamido]oxane-4-carboxylic acid
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(diethylamino)-3-[2-methoxy-5-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-[1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1H-pyrazol-4-yl]furan-2-carboxamide
N-ethyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-indole-7-carboxamide
2-(naphthalen-2-yloxy)-N-(oxan-4-yl)propanamide
4-(2,4-difluorophenyl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-ethyl-4-(4-ethylpiperazine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-methoxypyrazine
5-{[3-(benzyloxy)-4-methoxyphenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-{1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperazine-2-carbonyl}morpholine
(1S,5R)-3-(5-acetylpyridin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1,4-dithiepan-6-amine
4-{[1-(2-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
2-{2-[1-(1-methanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]phenoxy}acetic acid
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
3-[(2-methoxyethyl)(methyl)amino]-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
N-(3,4-dimethylphenyl)-2-{methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}acetamide
N-{4-[6-(dimethylamino)pyrimidin-4-yl]phenyl}-2-methylpropanamide
2-(4-methoxy-3,5-dimethylphenyl)-2-[methyl({2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})amino]acetic acid
(3S,4S)-4-propyl-1-[3-(pyridin-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
N-cyclopropyl-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(2-methoxyphenyl)methyl]benzamide
2,4-dichloro-3-({4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
1-[(3-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-chlorophenyl)-5-methyl-4-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperazin-2-one
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1,3-dimethyl 5-{[(1-methyl-6-oxopiperidin-3-yl)carbamoyl]amino}benzene-1,3-dicarboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-methyl-5-phenyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methoxyphenol
(3R,4R)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]propan-1-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl]urea