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(1S)-1-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]-2-phenylethan-1-ol
2-chloro-N-{[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]methyl}benzamide
N-(1-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
8-(2-ethylpyrimidine-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]piperidine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}propanamide
N-(6-phenoxypyridin-3-yl)-1-(thiophene-3-carbonyl)piperidine-4-carboxamide
N-butyl-N-methyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-(4-chloro-2-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}phenoxy)acetamide
1-(1H-1,3-benzodiazole-5-carbonyl)-4-hydroxypiperidine-4-carboxylic acid
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
2-(2-hydroxyethyl)-6-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-3-(4H-1,2,4-triazol-4-yl)propanamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpropanamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[2-(propylsulfanyl)phenyl]urea
4-amino-5-(1H-imidazol-2-yl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
2-(4-chloro-2-methylphenoxy)-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
3-(1-butyl-1H-pyrazol-5-yl)-1-[1-(thiophene-2-carbonyl)piperidin-3-yl]urea
4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-[1-(propan-2-yl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-methyl-3-(piperidin-4-ylmethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](cyclohexylmethyl)methylamine
N-[2-(1H-imidazol-4-yl)ethyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-[1-(2-methoxyphenoxy)propan-2-yl]pyrimidin-4-amine
2-fluoro-N-{3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}benzamide
3-[1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)pyrrolidin-2-yl]pyridine
2-benzyl-9-(3-hydroxypyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazole-2-carboxamide
9-(6-methylpyridazin-3-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-phenylpropan-2-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
[(2-methoxypyrimidin-5-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}thiophen-2-yl)ethan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
4-[(4-fluorophenyl)methyl]-1-[(4-hydroxyphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(pyridin-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]quinoline-4-carboxamide
(3E)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)pent-3-enamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
1-[2-methoxy-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydroquinoxalin-2-one
ethyl 3-(2-phenoxyethyl)-1-(pyrazine-2-carbonyl)piperidine-3-carboxylate
N-cycloheptyl-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propanamide
2-(3-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
4-[(2-methoxypyrimidin-5-yl)methyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
3-(2-fluorophenyl)-N-[(3-methylpyridin-4-yl)methyl]-3-phenylpropanamide
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-(2-chlorophenyl)piperazin-2-one