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(3R,4R)-4-(hydroxymethyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-ol
2-(2-hydroxyethyl)-9-(2,4,6-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,5-dimethyl-1H-indole-2-carboxamide
3-{[(1-methylpyrrolidin-3-yl)methyl]carbamoyl}adamantan-1-yl acetate
(4aR,8aR)-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-2H-1,4-benzoxazine
N-(1,2-oxazol-3-ylmethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-N-methylpiperidine-2-carboxamide
8-[(3-ethoxy-4-methoxyphenyl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(5-chlorothiophen-2-yl)methyl]-3-(2-methoxyphenoxy)azetidine
2-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-3-carboxamide
3-{[1-benzyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-(1-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
N-{1-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]piperidin-4-yl}methanesulfonamide
5-acetyl-N-[(4-methoxyphenyl)methyl]-N-propylthiophene-2-carboxamide
1-(2-ethoxyethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N'-(2-ethoxyphenyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylpropanediamide
2-{4-[(2,5-difluorophenyl)methyl]piperazin-1-yl}-N-ethyl-N-methylpyrimidin-4-amine
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(8-methoxyquinolin-2-yl)methyl]methylamine
4-[(2S)-2-hydroxy-3-phenylpropanoyl]-1-(2-methoxyphenyl)piperazin-2-one
3-({5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)propanamide
{4-[(4-methoxyphenyl)methyl]-1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}methanol
2-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]pyrazine
2,6,8-trimethyl-N-[(3S)-2-oxoazepan-3-yl]quinoline-4-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]oxane-4-carboxamide
2-[9-(2-methoxy-2-phenylacetyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
4-cyano-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrrole-2-carboxamide
2-(3-methoxypropyl)-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-1-yl}-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
6-cyclopentyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3aR,6aS)-5-[2-(1H-1,3-benzodiazol-2-ylmethoxy)acetyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
1-[(4-phenylphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
(3R,4R)-1-cyclobutanecarbonyl-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-3-ol
1-[(5-ethylpyridin-2-yl)methyl]-4-(4-fluorophenyl)piperazine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-6-hydroxy-N-methylpyridine-3-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}propan-1-one
3,7-dimethyl-11-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-3,7,11-triazaspiro[5.6]dodecane
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
1-(4-{[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidin-1-yl)ethan-1-one
2-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}-N-methylpentanamide
3-{1-[2-(2-hydroxyphenoxy)acetyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-4-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-{[3-(pyridin-2-yl)azetidin-1-yl]sulfonyl}morpholine
2-(dimethyl-1,3-thiazol-5-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylacetamide
N,N-dimethyl-N'-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanediamide
4-(cyclopropylmethyl)-1-(4-hydroxy-3-methoxybenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
3-(2,5-dihydroxy-2-methylpentyl)-1-[4-(4-methoxyphenyl)phenyl]urea
5-[1-(4-methanesulfonylphenyl)cyclohexyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(4-ethylpiperazin-1-yl)-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propan-1-one