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4-[2-(morpholin-2-yl)acetamido]-N-phenylpiperidine-1-carboxamide
1-[4-(1H-pyrazol-3-yl)phenyl]cyclopentane-1-carbonitrile
{6-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]pyridin-2-yl}methanol
4-[(2-fluorophenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
5,6-dimethyl-2-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-1,3-benzodiazole
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[2-(1H-pyrazol-1-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
methyl 6-(2-chlorobenzoyl)-2-(diethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-1-{2-[(3,5-dimethylphenyl)formamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(6-methylpyridin-2-yl)methyl]amine
[2-(3,5-dichlorophenyl)-1,3-thiazol-4-yl]methanol
3-(1-methyl-1H-pyrazol-4-yl)-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propan-1-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
2-(3-methoxy-4-methylphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
N-{2-[(6,6-dimethyl-5-oxothiomorpholin-3-yl)formamido]ethyl}pyridine-3-carboxamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4-diazepan-2-one
3-({2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
4-({1-benzyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1λ6-thiomorpholine-1,1-dione
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-ethyl-N,N-dimethyl-6-(4-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-propylpiperidin-4-amine
3-({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
3-chloro-5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
1-(2,2-dimethylpropyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-cyclopropyl-9-(1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-oxo-2-(thiophene-3-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(3-methoxyphenyl)methyl]acetamide
(1R,5S,6R,7S)-N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-propyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)piperidin-4-ol
1-{2-[1-(3-chloro-2-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
1-[2-(2,3-dihydro-1-benzofuran-7-yl)pyridine-4-carbonyl]-4-methylpiperazine
{[2-(difluoromethoxy)phenyl]methyl}({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
1-cyclopentyl-3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-(furan-2-ylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
2-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidin-1-yl}acetamide
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl][1-(2-fluorophenyl)propan-2-yl]amine
3-{[1-(pent-4-enoyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
(2S,4S)-4-amino-N-ethyl-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidine-2-carboxamide
N5-(1-benzylpiperidin-4-yl)-1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-fluoropyridine
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(cyclopent-1-ene-1-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole