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N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
1-[(4-methyl-1,3-thiazol-5-yl)methyl]azonan-2-one
{3-[(3-methoxyphenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methanol
methyl 4-{4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}benzoate
(1R,5R)-6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-N,N-dimethylaniline
1-cyclohexyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
3-(azocan-1-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(pyridin-4-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperazin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
methyl 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-ethyl-1H-pyrazole-5-carboxylate
1-ethyl-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-[methyl({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]propanamide
N-methyl-3-(3-methylpiperidin-1-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
4-{3-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]phenyl}-2-methylpyrimidine
2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-{4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-oxobutyl}pyrrolidin-2-one
(2R,3R)-3-[4-(ethanesulfonyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazole
4,6-dimethyl-1-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-(4-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}phenyl)acetamide
1-({2-[5-methyl-6-oxo-4-(trifluoromethyl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)piperidine-4-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(furan-2-yl)phenyl]-N-methylpiperidin-4-amine
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
3-(2-fluorophenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
[(5-chlorothiophen-2-yl)methyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
1-[(5-chlorofuran-2-yl)methyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
3-(2-hydroxyphenyl)-N-[4-methoxy-2-(2-methylpropanamido)phenyl]-1H-pyrazole-5-carboxamide
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
[(3aS,6aS)-2-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
methyl[(3-methylpyridin-2-yl)methyl]{[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
3-[(methylsulfanyl)methyl]-5-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole
2-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-({7-[4-(furan-2-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
1-{4-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-(3-chloro-4-methoxyphenyl)-2-(pyrrolidin-3-yl)benzamide
3-{[(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)oxy]methyl}pyridine
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
8-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-[3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanamido]acetate
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3R,4R)-3-hydroxy-1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide