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N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]propanamide
1-[2-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
8-(1-ethyl-1H-1,2,4-triazol-5-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(4aR,7aS)-1-[2-({imidazo[1,2-a]pyridin-2-ylmethyl}amino)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methoxy-3-[5-(morpholine-4-carbonyl)pyridin-2-yl]quinoline
2-{4-[(2-ethoxyphenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyridine-2-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-methoxypyrimidine-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-yl]pyridine-2-carboxamide
6-[(diethylamino)methyl]-N-[1-(4-fluorophenyl)ethyl]-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-ethoxy-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
4-(5-methylpyridin-2-yl)-1-(pyrazine-2-carbonyl)piperidin-4-ol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1-[(4-methoxyphenyl)amino]cyclopentane-1-carboxamide
2-ethoxy-6-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
5-ethyl-1'-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-4-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,3-thiazole-5-carboxamide
5-ethyl-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-cycloheptyl-2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]acetamide
3-(2-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
(1S,5R)-3-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[1-(methoxymethyl)cyclopentyl]-3-propyl-1H-pyrazole-5-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carbonitrile
1-(2,5-dimethylfuran-3-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
6-cyclopropyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]pyrimidin-4-amine
4-[5-(5-methylpyrazin-2-yl)-1,2,4-oxadiazol-3-yl]-1H-indole
N-[2-(diethylamino)ethyl]-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridine-2-carboxamide
5-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-(4-methoxy-2-methylphenyl)-3-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}propanamide
4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}benzonitrile
N-(3-hydroxypropyl)-3-(methylsulfanyl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
1-(2-amino-9H-purin-6-yl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
4-(2,3-dihydro-1-benzofuran-5-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(morpholin-4-yl)pentan-1-one
ethyl 2-(4-{2-[4-(furan-2-amido)-1H-pyrazol-1-yl]acetyl}morpholin-3-yl)acetate
1-(cyclopropylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethyl-1,2-oxazol-4-yl)-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]acetamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-(4-fluorophenyl)-6,6-dimethyl-N-(1-methylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
{1-[3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propyl]piperidin-2-yl}methanol
5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-ethyl-2-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,3-thiazole-5-carboxamide