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(3R,4R)-1-cyclobutanecarbonyl-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-hydroxy-N,2-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-5-carboxamide
5-[1-({2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-4-yl}methyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(propan-2-yl)-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
3-methoxy-2,2-dimethyl-N-{1-[2-(trifluoromethyl)phenyl]ethyl}propanamide
2-acetyl-8-(4-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propan-1-one
3-(3-chloro-4-ethoxyphenyl)-1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
{1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
methyl 3-(cyclobutylmethoxy)-5-(1,4-oxazepane-4-carbonyl)benzoate
(3S,4R)-1-[(6-chloro-2H-chromen-3-yl)methyl]-4-methylpiperidine-3,4-diol
3-[(3-carbamoylphenyl)methyl]-N-(2-ethoxyphenyl)pyrrolidine-1-carboxamide
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
4-(1,4-oxazepan-4-ylmethyl)quinoline
9-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-[(4-fluorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
methyl 1-{[4-(3,4-difluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
2-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
N-[2-ethyl-4-(8-methoxyquinolin-5-yl)phenyl]acetamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-{1-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
7-[(2R)-2-amino-3-(ethylsulfanyl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(3-chloro-2-ethoxyphenyl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
N-{2-[4-({[(2-butyl-1H-imidazol-4-yl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide
N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
1-(2-ethoxyethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-(thiomorpholin-4-yl)propan-1-one
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
1-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[(4-fluorophenyl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
7-(2,5-dimethylfuran-3-carbonyl)-2-[(2E)-hex-2-en-1-yl]-2,7-diazaspiro[4.5]decane
7-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-methyl-4-({5-[(2-phenyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
3-(oxolan-3-yl)-5-(1-phenylcyclopentyl)-1,2,4-oxadiazole
8-[(3-methoxyphenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-{3-[({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)amino]-2-methylphenyl}-3-methylbutanamide
4-(2,6-dimethylpyridin-3-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
2-(3-fluorophenyl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide