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2-(5-methyl-1H-pyrazol-1-yl)-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
5-methoxy-2-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridin-4-ol
1-[3-({3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
1-{3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}propan-1-one
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-3-(1H-imidazol-2-yl)benzamide
methyl 2-[4-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2-oxopiperazin-1-yl]acetate
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
1-ethyl-3-methyl-4-(2-phenylpyrrolidine-1-carbonyl)-1H-pyrazole
1,2-dimethyl-4-{[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}-1H-imidazole
N-methyl-5-{[methyl(2-phenoxyethyl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)piperidin-2-one
N-[2-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)ethyl]acetamide
3-chloro-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyrrolidin-1-yl)benzamide
2-cyclopropyl-5-{1-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}pyrimidine
N-[3-(azepan-1-yl)propyl]-N,4,6-trimethylpyrimidin-2-amine
3-(dimethyl-1,2-oxazol-4-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
1-(4-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-cyclohexyl-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidine
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-methoxy-4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoline
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}ethan-1-one
2-(ethylamino)-N-[(4-fluorophenyl)methyl]-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-[2-(dimethylamino)ethyl]-5-(3-methylpyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(3-methylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,8aR)-1-(3-methoxypropyl)-6-(1-phenylpiperidin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-(4-fluorophenyl)-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-one
1-[(4-fluoro-3-methylphenyl)methyl]-3-[3-(piperidine-1-carbonyl)phenyl]urea
N-(4-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanamido}-2-methoxyphenyl)butanamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
2-(2-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-fluoro-3,4-dihydroquinazolin-4-one
2-(2-phenyl-1,3-thiazol-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(3-hydroxypropyl)piperidine-3-carboxamide
N-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(thiophene-2-carbonyl)piperidin-3-amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
2-(4-chlorophenyl)-4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]morpholine
2-[benzyl({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
methyl (2R,4S)-1-(4-chloro-2,5-dimethylbenzenesulfonyl)-4-hydroxypiperidine-2-carboxylate
3-methyl-4-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-propyl-1H-pyrazole
2-({[1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-{4-[({[1-(ethoxymethyl)cyclobutyl]methyl}carbamoyl)methoxy]phenyl}propanamide
2-methyl-8-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-2,8-diazaspiro[5.5]undecane
(2R,6R)-10-methoxy-4-(morpholine-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
1-(3-chlorophenyl)-4-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine