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(3R,5S)-N-[2-(dimethylamino)ethyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-ethyl-3-[1-(2-{3-methyl-2-oxo-2H,3H-imidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 1-({6-[methyl(2-phenylethyl)carbamoyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-4-carboxylate
5-(3-methylbutyl)-3-[2-(2-oxopyrrolidin-1-yl)ethyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-(benzyloxy)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
6-[4-(methoxymethyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(thian-4-yl)piperazine
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-pyrrole-2-carboxamide
3-[(2-ethylpiperidin-1-yl)methyl]-7-fluoro-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-2-one
1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
1-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]urea
1'-(2,6-dimethylpyridin-4-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-(4-methyl-1H-pyrazol-3-yl)-1-(oxolan-3-ylmethyl)piperidine
1-[1'-(4-ethenylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-[methyl({2-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl})amino]-1λ6-thiolane-1,1-dione
1-(2-methyl-1H-imidazole-4-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
(2,3-dihydro-1-benzofuran-5-ylmethyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
4-(1,2,3,4-tetrahydronaphthalen-1-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1,5-dimethyl-4-{[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]methyl}-1H-pyrrole-2-carbonitrile
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
2,3,5-trimethyl-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(3-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
N-(2,2-difluoroethyl)-4-[3-(hydroxymethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-({[(4-chlorophenyl)methyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
N,7-bis(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-chloro-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
1-[(2-chloro-6-fluorophenyl)methyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-7-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline
3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}phenol
(1R,5R)-6-(cyclobutylmethyl)-3-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{2-chloro-4-[1-(2-methylpropyl)-1H-imidazol-2-yl]phenoxy}acetamide
1-ethyl-3-(2-methylpropyl)-N-[(2,3,6-trifluorophenyl)methyl]-1H-pyrazole-5-carboxamide
2-({4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
1-(3-fluoropyridin-2-yl)-4-(thian-4-yl)piperazine
N-cyclobutyl-2-(2-methylpentanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
{1-[(6-fluoroquinolin-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
1-[2-(3-chloro-4-methoxyphenyl)pyrimidin-4-yl]piperidin-4-ol
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-ethyl-3-methyl-N-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}aniline
1-(diphenylmethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-(3-fluorophenyl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-{[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-(3-methylphenyl)piperazine
N-(cyclohex-1-en-1-ylmethyl)-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
1-{[4-(3-ethylphenoxy)-3-methoxyphenyl]methyl}pyrrolidine